Target Details
| UniProt AC | P48546 |
|---|---|
| Gene Symbol | GIPR |
| Protein Name | Gastric inhibitory polypeptide receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 96
- Clinical molecules 0
- Avg pChEMBL 6.68
KEGG Pathways (3)
Active Molecules (96)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SLYYRVVPLWMNPO
|
6.4 | IC50 | 2 | — | |
SYWXLIGCTNVJDM
|
6.4 | IC50 | 2 | — | |
YAJKYUVXRYCKPC
|
6.4 | IC50 | 2 | — | |
FVDONABKZHMTCY
|
6.4 | IC50 | 2 | — | |
HHKKVYXTKFAECF
|
6.4 | IC50 | 2 | — | |
JTMDOZVHCVTETN
|
6.4 | IC50 | 2 | — | |
NPMZBYQQJWHAEW
|
6.4 | IC50 | 2 | — | |
XNSJRSAITGCUKS
|
6.3 | IC50 | 2 | — | |
VEXHFZLCFRSPSZ
|
6.3 | IC50 | 2 | — | |
SVLDQMHFIWDPJO
|
6.3 | IC50 | 2 | — | |
MYHQPEVOOWDUDW
|
6.3 | IC50 | 2 | — | |
OTDAFCWROVFKOL
|
6.3 | IC50 | 2 | — | |
OTDAFCWROVFKOL
|
6.3 | IC50 | 2 | — | |
WFUXVTIXEWVFED
|
6.3 | IC50 | 2 | — | |
BKFPJEBZTCJJRP
|
6.3 | IC50 | 2 | — | |
NGUABMKOSJANPJ
|
6.2 | IC50 | 2 | — | |
SGTLXOZGCVZYAN
|
6.2 | IC50 | 2 | — | |
FDAPJZJLEIYQAN
|
6.2 | IC50 | 2 | — | |
KNMAVSXEMFMOGI
|
6.2 | IC50 | 2 | — | |
MTBJTQZAQADZQL
|
6.2 | IC50 | 2 | — | |
MDDANNKYTHKAHR
|
6.2 | IC50 | 2 | — | |
MYYKZRMEYNXGOG
|
6.2 | IC50 | 2 | — | |
GKFODRKFKVOWTH
|
6.2 | IC50 | 2 | — | |
KOVJJWYJLGKJAI
|
6.2 | IC50 | 2 | — | |
GLTBMLMTGHGENX
|
6.2 | IC50 | 2 | — | |
XNSJRSAITGCUKS
|
6.2 | IC50 | 2 | — | |
CTOLIBJXQJXWDY
|
6.1 | IC50 | 2 | — | |
WPHHXNCBGPKNOY
|
6.1 | IC50 | 2 | — | |
XKENBIHIHWFSFY
|
6.1 | IC50 | 2 | — | |
KNTOEHKTBLUGLN
|
6.1 | IC50 | 2 | — | |
YQWKQQFUAPWMJC
|
6.1 | IC50 | 2 | — | |
XKURAAGCCZEBHF
|
6.1 | IC50 | 2 | — | |
ICARRUHVPUOWDW
|
6.1 | IC50 | 2 | — | |
HHLCSKJKCZOHTH
|
6.1 | IC50 | 2 | — | |
VDRBYJICTVBZID
|
6.1 | IC50 | 2 | — | |
XEECUIDWJQYSIO
|
6.1 | IC50 | 2 | — | |
ITDOIINIFNQSFX
|
6.0 | IC50 | 2 | — | |
QGUIDVPVMJAYTK
|
6.0 | IC50 | 2 | — | |
RSJWMKGJEAKNNJ
|
6.0 | Ki | 2 | — | |
UXPYCHMVTKGDJP
|
6.0 | IC50 | 2 | — | |
VERXBCYVZFLZNT
|
6.0 | Ki | 2 | — | |
YZUIGWQMHIUXNA
|
6.0 | IC50 | 2 | — | |
CTJDFSIKSQVUTF
|
6.0 | IC50 | 2 | — | |
CWPADRJBQLPUCB
|
6.0 | IC50 | 3 | — | |
FTBIQPJNXCTJIU
|
6.0 | IC50 | 2 | — | |
WCVRCGUPWLUXJR
|
6.0 | IC50 | 2 | — |