Target Details
| UniProt AC | P48546 |
|---|---|
| Gene Symbol | GIPR |
| Protein Name | Gastric inhibitory polypeptide receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 96
- Clinical molecules 0
- Avg pChEMBL 6.68
KEGG Pathways (3)
Active Molecules (96)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QADDVLGUGQIQSK
|
9.8 | IC50 | 2 | — | |
LVHVRGDXLSIEGE
|
9.1 | IC50 | 2 | — | |
YRJNFJTUXZVAHI
|
9.0 | IC50 | 2 | — | |
JOEIAOIUXPYGIF
|
9.0 | IC50 | 2 | — | |
AYEQXACAEGGPLJ
|
8.9 | IC50 | 2 | — | |
FYZOUIJJKZBMFX
|
8.6 | IC50 | 2 | — | |
OXFQTDZOCZPPCB
|
8.3 | IC50 | 2 | — | |
REIGIHUHXDNPSA
|
7.9 | IC50 | 2 | — | |
NCTZKXFEIKKURA
|
7.9 | IC50 | 2 | — | |
BZXMLCVDKDXRQY
|
7.5 | IC50 | 2 | — | |
POXYYUCJPKWULA
|
7.4 | IC50 | 2 | — | |
WGMDTVFTELHPOL
|
7.4 | IC50 | 2 | — | |
VSGDYFXFEPKTGU
|
7.3 | IC50 | 2 | — | |
QVSVLRYVPXFJOT
|
7.2 | IC50 | 3 | — | |
VHURVYZHODPCCB
|
7.2 | IC50 | 2 | — | |
AKFRCBAYXPRXSG
|
7.1 | IC50 | 2 | — | |
SPYNVKYBDKGKEH
|
7.1 | IC50 | 2 | — | |
OIQWAEIGTZYWRX
|
7.1 | IC50 | 2 | — | |
DAUDLQFCWWLQPT
|
7.0 | IC50 | 2 | — | |
MRJZJRLNCMMRCZ
|
7.0 | IC50 | 2 | — | |
OLGWNKHCHXVJMX
|
7.0 | IC50 | 2 | — | |
SQCUILFEAKKVAC
|
6.9 | IC50 | 2 | — | |
XTOBAVZIBVVXLS
|
6.9 | IC50 | 2 | — | |
KNMAVSXEMFMOGI
|
6.9 | IC50 | 2 | — | |
KOZDDXIYVDHLIC
|
6.8 | IC50 | 2 | — | |
VOSMSHCJSJBJOD
|
6.8 | IC50 | 2 | — | |
CHYPABFSTPTACZ
|
6.8 | IC50 | 2 | — | |
ANMUHQCUTMTNRH
|
6.7 | IC50 | 2 | — | |
OUZOYODGROMRMW
|
6.7 | IC50 | 2 | — | |
QJEGIIJPDLHOEZ
|
6.7 | IC50 | 2 | — | |
QCXYVMFKAJYFNH
|
6.7 | IC50 | 2 | — | |
VLGOFRLXSHLEAO
|
6.7 | IC50 | 2 | — | |
YDAXDTSMRRYDQR
|
6.6 | IC50 | 2 | — | |
JKDNPQJPEAQBPC
|
6.5 | IC50 | 2 | — | |
LOKUGNIDKBRXJC
|
6.5 | IC50 | 2 | — | |
LOKUGNIDKBRXJC
|
6.5 | IC50 | 2 | — | |
YXRLENJRMMVUDH
|
6.5 | IC50 | 2 | — | |
NPMZBYQQJWHAEW
|
6.5 | IC50 | 2 | — | |
ZBMZGBGZOQFXEP
|
6.5 | Ki | 3 | — | |
QLCNDVIJFAHAFO
|
6.5 | IC50 | 2 | — | |
CIDYLAWHEXYTGX
|
6.5 | IC50 | 2 | — | |
DRBYFBHVRFFBIU
|
6.5 | IC50 | 2 | — | |
XNSJRSAITGCUKS
|
6.4 | IC50 | 2 | — | |
BOPMXYXKSFCVIW
|
6.4 | IC50 | 2 | — | |
OIQWAEIGTZYWRX
|
6.4 | IC50 | 2 | — | |
UECFQNMLGNHNSO
|
6.4 | IC50 | 2 | — | |
UECFQNMLGNHNSO
|
6.4 | IC50 | 2 | — | |
MYFXPJIUHYQWRX
|
6.4 | IC50 | 2 | — | |
OBRBSPYTOYTECA
|
6.4 | IC50 | 2 | — | |
QMZREIRRGCJPTH
|
6.4 | IC50 | 2 | — |