Target Details
| UniProt AC | P48454 |
|---|---|
| Gene Symbol | PPP3CC |
| Protein Name | Serine/threonine-protein phosphatase 2B catalytic subunit gamma isoform |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00149 (Metallophos) |
Summary
- Multi-target molecules 27
- Clinical molecules 0
- Avg pChEMBL 6.61
KEGG Pathways (33)
- Alzheimer disease
- Amphetamine addiction
- Amyotrophic lateral sclerosis
- Axon guidance
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Calcium signaling pathway
- Cellular senescence
- Dopaminergic synapse
- Glucagon signaling pathway
- Glutamatergic synapse
- Human T-cell leukemia virus 1 infection
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Long-term potentiation
- MAPK signaling pathway
- Natural killer cell mediated cytotoxicity
- Oocyte meiosis
- Osteoclast differentiation
- Oxytocin signaling pathway
- PD-L1 expression and PD-1 checkpoint pathway in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Renin secretion
- T cell receptor signaling pathway
- Th1 and Th2 cell differentiation
- Th17 cell differentiation
- Tuberculosis
- VEGF signaling pathway
- Wnt signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMGVCDCNHBXLNW
|
7.3 | IC50 | 2 | — | |
QNOPKSIUIKQNNW
|
7.1 | IC50 | 2 | — | |
SOLUUOZSPTULAB
|
7.1 | IC50 | 2 | — | |
GPFMVNBJTPRJJI
|
6.9 | IC50 | 2 | — | |
YJQKYLZBYOCLDJ
|
6.9 | IC50 | 2 | — | |
PJFCXNVGTPNOPO
|
6.8 | IC50 | 2 | — | |
RGTWDGJFJKIHQZ
|
6.7 | IC50 | 2 | — | |
GJKSJDQWTGQEAL
|
6.7 | IC50 | 2 | — | |
PMATZTZNYRCHOR
|
6.7 | IC50 | 20 | — | |
QQJWZNXLWRBBHE
|
6.7 | IC50 | 2 | — | |
VWILXAVJHMPMLD
|
6.7 | IC50 | 2 | — | |
UQPPGSWGYIDVBM
|
6.6 | IC50 | 2 | — | |
IIJBDKQYIBVJEJ
|
6.6 | IC50 | 2 | — | |
FWOMHUCZELGHDG
|
6.5 | IC50 | 2 | — | |
XEVOFZMUTYYQEF
|
6.5 | IC50 | 2 | — | |
YXTRRTPUHABKMO
|
6.5 | IC50 | 2 | — | |
AVGTWAFRISPNPD
|
6.5 | IC50 | 2 | — | |
CFLIZBNNTWMZBS
|
6.5 | IC50 | 2 | — | |
PWUIJAMDQQVCRY
|
6.5 | IC50 | 2 | — | |
LWNMJUSNWZCTRX
|
6.5 | IC50 | 2 | — | |
JDJHHVLRQBGILF
|
6.4 | IC50 | 2 | — | |
KQWBVYSVPDFJBS
|
6.4 | IC50 | 2 | — | |
FUXQCGDBZUJIMC
|
6.4 | IC50 | 2 | — | |
KEIAKVUMZMYHRT
|
6.4 | IC50 | 2 | — | |
PSMUBOWUHXAYOX
|
6.3 | IC50 | 2 | — | |
GSWMITGBVBPMIW
|
6.3 | IC50 | 2 | — | |
RZVOFVMPJWTZOT
|
6.2 | IC50 | 2 | — |