Target Details
| UniProt AC | P48169 |
|---|---|
| Gene Symbol | GABRA4 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 364
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (8)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DQDLJDCSJFQOHI
|
6.0 | IC50 | 16 | — | |
FKRRGAJQEMJONC
|
6.0 | Ki | 7 | — | |
FUULVCWWUPGUMY
|
6.0 | IC50 | 16 | — | |
FVFFDKKTXYVCCW
|
6.0 | Ki | 16 | — | |
GCTOZKWOFVUEAW
|
6.0 | IC50 | 16 | — | |
IHFBPDAQLQOCBX
|
6.0 | Ki | 18 | — | |
KBMIXEOSQPPORV
|
6.0 | Ki | 8 | — | |
KVZVPZYFPDOIMI
|
6.0 | IC50 | 16 | — | |
LPAODQAWVMEXKR
|
6.0 | Ki | 16 | — | |
LTYUPBZLKIUGQX
|
6.0 | Ki | 8 | — | |
OSMYMXKHKOTLKC
|
6.0 | Ki | 7 | — | |
RYFIWEJRWHTFBM
|
6.0 | IC50 | 16 | — | |
SIPHVHFVEKBHKT
|
6.0 | Ki | 7 | — | |
TTXJJFWWNDJDNR
|
6.0 | IC50 | 3 | — |