Target Details
| UniProt AC | P48169 |
|---|---|
| Gene Symbol | GABRA4 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 364
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (8)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DNCFKDLZZSXXJP
|
6.4 | IC50 | 16 | — | |
MUPIUJYENVWEKT
|
6.4 | IC50 | 16 | — | |
NQFQEBQBZXSXIX
|
6.4 | IC50 | 16 | — | |
QYSYOGCIDRANAR
|
6.4 | Ki | 7 | — | |
VNFZCRPFALLSNM
|
6.4 | IC50 | 16 | — | |
SQPWTARSPNZNEI
|
6.4 | IC50 | 16 | — | |
QCSFXCHHKYXLHE
|
6.4 | Ki | 16 | — | |
YFEZLTPSCJWVHI
|
6.4 | Ki | 16 | — | |
YOJAHANNNITYMX
|
6.4 | Ki | 16 | — | |
ZLAPTIDQRXJQQL
|
6.4 | IC50 | 16 | — | |
AEPFXRGRJZMVIF
|
6.3 | Ki | 17 | — | |
JBTLCAMUYYCXTA
|
6.3 | IC50 | 16 | — | |
DKCNNHVHQYMVTO
|
6.3 | IC50 | 16 | — | |
BDGWCPYUERFMMY
|
6.3 | Ki | 16 | — | |
UMYWGMKUCZAQJO
|
6.3 | Ki | 16 | — | |
FNZFELZOBRBQJY
|
6.3 | IC50 | 16 | — | |
IGCSLIVTBUKKRS
|
6.3 | IC50 | 16 | — | |
SRJOCJYGOFTFLH
|
6.3 | Ki | 16 | — | |
IKDYRDIWKFJQTR
|
6.3 | IC50 | 16 | — | |
PZWMQJZDDYQYGN
|
6.3 | Ki | 16 | — | |
ZEEOGWVZWOURAE
|
6.2 | Ki | 16 | — | |
OMGOVFIKWLKTPS
|
6.2 | Ki | 16 | — | |
BZIBRALMCDHACX
|
6.2 | Ki | 17 | — | |
JWTQJUQJIRWZLA
|
6.2 | Ki | 16 | — | |
ODWCGGCCGLKRAK
|
6.2 | Ki | 16 | — | |
ICRYUJPBYIPXQF
|
6.2 | IC50 | 16 | — | |
ZMKDYQONTIIETL
|
6.2 | Ki | 16 | — | |
OJOTYQLMNVPQBO
|
6.2 | Ki | 16 | — | |
RRAXPPHKWFOGGL
|
6.2 | Ki | 16 | — | |
WQIWYEISPHMPOA
|
6.2 | IC50 | 16 | — | |
ARCJBXYEOMXBSZ
|
6.2 | IC50 | 16 | — | |
CTPREUOHTKHCHT
|
6.2 | IC50 | 16 | — | |
KOVRZNUMIKACTB
|
6.2 | Ki | 17 | — | |
XFUAEWGHLXLENC
|
6.2 | IC50 | 16 | — | |
BSEVRQDRIQMBCV
|
6.2 | IC50 | 16 | — | |
DHEXTYZLLGWEFS
|
6.2 | Ki | 16 | — | |
HBOSSQBJUBOEJN
|
6.1 | Ki | 16 | — | |
XVFJUDUNNHPHLN
|
6.1 | IC50 | 16 | — | |
HYJUIJYNZHZBOK
|
6.1 | IC50 | 16 | — | |
WJEPRNMCEBRSDB
|
6.1 | IC50 | 16 | — | |
YLZBNNDOEUIHFB
|
6.1 | IC50 | 16 | — | |
LKUSWPRPRBXYPH
|
6.1 | IC50 | 16 | — | |
VKMJGKFQKLVODR
|
6.1 | IC50 | 16 | — | |
VAEZVMCCCWEXEH
|
6.1 | Ki | 16 | — | |
ZXYMHGABHZSFOI
|
6.1 | Ki | 16 | — | |
DOOGDICMBOTQOZ
|
6.1 | IC50 | 16 | — | |
SLNCMJYPLFSUGO
|
6.0 | Ki | 16 | — | |
SZHSENNQOQSFEA
|
6.0 | IC50 | 16 | — | |
ACHPNNOYBNCORU
|
6.0 | Ki | 8 | — | |
DHLJRIFIBJGWBS
|
6.0 | IC50 | 16 | — |