Target Details
| UniProt AC | P48169 |
|---|---|
| Gene Symbol | GABRA4 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 364
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (8)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XAXZXMJZHNVJEQ
|
6.8 | Ki | 16 | — | |
CGOOGLSJSVATGZ
|
6.8 | Ki | 16 | — | |
FLHRNVLCKMTQAP
|
6.8 | Ki | 17 | — | |
JQHJWKNJYLNAFL
|
6.8 | IC50 | 16 | — | |
DLEWDNHPWLPKDJ
|
6.8 | Ki | 8 | — | |
FCBAIIQUIRAZRU
|
6.8 | Ki | 4 | — | |
XLKFCRQJPWBJNW
|
6.8 | IC50 | 16 | — | |
CGVJPQYHXQIFPE
|
6.7 | Ki | 16 | — | |
PGTVWKLGGCQMBR
|
6.7 | IC50 | 16 | — | |
QKZNNAUSAVZXNE
|
6.7 | Ki | 16 | — | |
HGPFVUUTSFNGNR
|
6.7 | Ki | 18 | — | |
FRKWUXZCSLOPIC
|
6.7 | IC50 | 7 | — | |
AYRJXCIMSHQLPG
|
6.7 | Ki | 6 | — | |
GMVMGIYPRPPNMB
|
6.7 | Ki | 16 | — | |
ZRKQHHNVLRRZFQ
|
6.7 | Ki | 16 | — | |
PTRPQDMPYNOBTR
|
6.7 | IC50 | 16 | — | |
DATCQVJMADOCRS
|
6.7 | IC50 | 16 | — | |
GXUSNZYZTBJMIT
|
6.7 | Ki | 16 | — | |
KNZNHUNBVIKNJP
|
6.7 | Ki | 5 | — | |
SINAJPKUKOSXOT
|
6.7 | IC50 | 16 | — | |
WFRRJMYHDPXXFB
|
6.7 | Ki | 16 | — | |
YWCLXVVWMQVKRF
|
6.7 | IC50 | 16 | — | |
CELFESKDAXZKDL
|
6.6 | IC50 | 16 | — | |
HXXGVDKGNHCARX
|
6.6 | IC50 | 16 | — | |
VMNYVCMDPUOQEL
|
6.6 | Ki | 16 | — | |
GXFWOMYQHNODFA
|
6.6 | IC50 | 16 | — | |
HOTHDLMXYUFPSZ
|
6.6 | IC50 | 16 | — | |
QQONDVXXMVPYIB
|
6.6 | Ki | 16 | — | |
YTGZSWOWFGVAFH
|
6.6 | Ki | 7 | — | |
GCNSLTKPBZQFJK
|
6.6 | IC50 | 16 | — | |
ODIZUHKZJZYZAL
|
6.6 | IC50 | 16 | — | |
RTMFRAUTYIKCRK
|
6.6 | Ki | 16 | — | |
WNDIDYSCZWXEJF
|
6.6 | Ki | 16 | — | |
LOBNIVNGRUTMOS
|
6.5 | IC50 | 16 | — | |
WRUTXEAYYQYJHO
|
6.5 | Ki | 16 | — | |
YTTJSPTYQMWSNO
|
6.5 | Ki | 5 | — | |
FXYDXLJEJBXFBD
|
6.5 | IC50 | 7 | — | |
HJGRBNHROFTASJ
|
6.5 | IC50 | 16 | — | |
QMCOPDWHWYSJSA
|
6.5 | Ki | 2 | — | |
YHZXFRGWTKYPKS
|
6.5 | Ki | 16 | — | |
GAQCKHAXURZXGX
|
6.5 | IC50 | 16 | — | |
UKHFPVCOXBJPIN
|
6.5 | Ki | 17 | — | |
VEWLYIAEUXDQBW
|
6.5 | IC50 | 16 | — | |
GDVGLPNNOCDLLD
|
6.5 | IC50 | 16 | — | |
GEFDSAOHFGLQEZ
|
6.5 | Ki | 17 | — | |
WCTCMHZWHMFZFN
|
6.5 | Ki | 17 | — | |
DDSULWHSYUPHBK
|
6.5 | IC50 | 16 | — | |
HARMZUHRUKGCNG
|
6.5 | Ki | 8 | — | |
XRWYYMUIIXMQBL
|
6.5 | IC50 | 16 | — | |
DAYQXLQRTQODQF
|
6.4 | Ki | 16 | — |