Target Details
| UniProt AC | P48169 |
|---|---|
| Gene Symbol | GABRA4 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 364
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (8)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NFXAWQDTYKJJTD
|
7.1 | IC50 | 16 | — | |
PQGDUNWRHHLMNT
|
7.1 | Ki | 9 | — | |
JSRKYARWMIOKOB
|
7.0 | Ki | 16 | — | |
LWLYOXPDYPYNHH
|
7.0 | IC50 | 16 | — | |
SZSNAHWJFCIUBV
|
7.0 | IC50 | 17 | — | |
WUNJCJOCGLXHNU
|
7.0 | IC50 | 16 | — | |
GSNCQRDETZIWAE
|
7.0 | Ki | 16 | — | |
KWHWSXISOMCUPZ
|
7.0 | IC50 | 16 | — | |
VDAHGXKTABYDOQ
|
7.0 | Ki | 16 | — | |
XJSZCKCJAMOVEP
|
7.0 | IC50 | 16 | — | |
OWUSBEXUSSJSDZ
|
7.0 | IC50 | 16 | — | |
HMRWJLKGQUMXKG
|
7.0 | IC50 | 9 | — | |
PWFUHHSGSJDKCU
|
7.0 | IC50 | 16 | — | |
XPRGZRFECLBYKZ
|
7.0 | IC50 | 9 | — | |
GBBSUAFBMRNDJC
|
7.0 | Ki | 6 | — | |
KQTMWRZAVOUNCI
|
7.0 | IC50 | 16 | — | |
DVKHCFDZNVGRQT
|
7.0 | IC50 | 16 | — | |
IIDOALWZHDFUQF
|
7.0 | IC50 | 16 | — | |
FQDQLHDSVITISC
|
7.0 | IC50 | 16 | — | |
YEFFWDGMWBFKHL
|
7.0 | Ki | 16 | — | |
RMGFIVKKLZZKNY
|
7.0 | IC50 | 16 | — | |
XVRONCOEBFKZEW
|
7.0 | IC50 | 16 | — | |
LUDMNXOOXWWZDU
|
6.9 | Ki | 7 | — | |
NMMJOCVBNVTBNP
|
6.9 | Ki | 16 | — | |
GQXSRHIFUJLCSW
|
6.9 | Ki | 16 | — | |
JYXHNHBKWZQGLB
|
6.9 | Ki | 16 | — | |
HWOWPGLTTSFLOQ
|
6.9 | Ki | 16 | — | |
OOAXMNBBGAIJCT
|
6.9 | Ki | 7 | — | |
VFKHADGYGKHTDK
|
6.9 | IC50 | 16 | — | |
LHSWKUZVAZKLHJ
|
6.9 | IC50 | 16 | — | |
VFPUCBWBLOQFPU
|
6.9 | IC50 | 16 | — | |
YZBJLGYBBNTKKL
|
6.9 | IC50 | 16 | — | |
VHBFFQKBGNRLFZ
|
6.9 | Ki | 21 | — | |
ACPUCHLYONVNTK
|
6.9 | Ki | 16 | — | |
VMDUABMKBUKKPG
|
6.9 | Ki | 16 | — | |
XYLGLGFZLQRDKD
|
6.9 | Ki | 16 | — | |
BIHMYZHWJAFHBO
|
6.8 | IC50 | 16 | — | |
KOTFZRCPKVQWPP
|
6.8 | Ki | 16 | — | |
XLKFCRQJPWBJNW
|
6.8 | IC50 | 16 | — | |
KTFRBKXLNKKPEA
|
6.8 | IC50 | 16 | — | |
DGWAMRKYNYINRJ
|
6.8 | IC50 | 16 | — | |
QQXJSYFEJVOQLZ
|
6.8 | IC50 | 16 | — | |
VGZQARXDBOOWBF
|
6.8 | Ki | 16 | — | |
GZGLGVQROXSNSN
|
6.8 | Ki | 9 | — | |
JTQDBIFZWJTIIQ
|
6.8 | Ki | 16 | — | |
JXKAURVNHHPPND
|
6.8 | IC50 | 16 | — | |
RHARCGZTSJROQQ
|
6.8 | Ki | 16 | — | |
RLKPTPBBRCFHEK
|
6.8 | IC50 | 16 | — | |
BXKSCEUJEPDZBI
|
6.8 | Ki | 16 | — | |
STQWWORVIGBLOE
|
6.8 | Ki | 16 | — |