Target Details
| UniProt AC | P48169 |
|---|---|
| Gene Symbol | GABRA4 |
| Protein Name | Gamma-aminobutyric acid receptor subunit alpha-4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 364
- Clinical molecules 0
- Avg pChEMBL 7.31
KEGG Pathways (8)
Active Molecules (364)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SCAPGUIFNHZJLH
|
7.5 | IC50 | 16 | — | |
SUONVKFDJJYYME
|
7.5 | IC50 | 16 | — | |
QJCQEAQHBMKTCT
|
7.5 | IC50 | 16 | — | |
LWUDDYHYYNNIQI
|
7.4 | Ki | 6 | — | |
DOKJHXYCSUQRQV
|
7.4 | Ki | 16 | — | |
JGVCISSLGASTTA
|
7.4 | Ki | 18 | — | |
FXIDXTIMKAEBGY
|
7.4 | Ki | 7 | — | |
GCSRDJACUSRHBX
|
7.4 | Ki | 16 | — | |
FXYDXLJEJBXFBD
|
7.4 | IC50 | 6 | — | |
CMVZUGQWJUPOJA
|
7.4 | IC50 | 16 | — | |
QMHTYKLXSOQULX
|
7.4 | Ki | 16 | — | |
DUZTVXKYJROMJJ
|
7.4 | IC50 | 16 | — | |
BMIKDIWICOAHJN
|
7.4 | Ki | 16 | — | |
MSFAMEBSEKIVDI
|
7.4 | Ki | 16 | — | |
VUZAUNZSDCMUTH
|
7.4 | Ki | 16 | — | |
LDBHRENGPXWKOD
|
7.3 | IC50 | 16 | — | |
GWCQPEHFUKZODL
|
7.3 | Ki | 16 | — | |
QYEIQYJLVREYBI
|
7.3 | IC50 | 16 | — | |
SIBRGSBVGDWJAF
|
7.3 | IC50 | 16 | — | |
WHGIBMIKSVYLCR
|
7.3 | IC50 | 16 | — | |
AURFZBICLPNKBZ
|
7.3 | IC50 | 16 | — | |
GQIVRYNNTCEOBX
|
7.3 | Ki | 8 | — | |
DGZYPGWWTKGBQP
|
7.3 | Ki | 16 | — | |
NTZNKZHCQIJCPO
|
7.3 | IC50 | 16 | — | |
SNEWVMXJSABDSK
|
7.3 | Ki | 16 | — | |
VWCCHJFFYCGXFL
|
7.3 | Ki | 16 | — | |
WDTNKNNGHGOKBH
|
7.3 | Ki | 9 | — | |
JBDRNSFDKSBSFE
|
7.3 | Ki | 16 | — | |
NNHRCSJWUBQYQV
|
7.3 | IC50 | 16 | — | |
PISRVNOAPOPQHJ
|
7.3 | Ki | 18 | — | |
KRVDMABBKYMBHG
|
7.3 | Ki | 16 | — | |
VOZOMZWSLGQRKP
|
7.3 | IC50 | 16 | — | |
XEJHLKHWRSNEOC
|
7.3 | IC50 | 16 | — | |
UEWSJGMYAPQKKT
|
7.2 | Ki | 16 | — | |
URMNROOZTOLUHQ
|
7.2 | Ki | 16 | — | |
PWOQCZLPANHRRJ
|
7.2 | Ki | 16 | — | |
NKSQLOHZBFUKLF
|
7.2 | IC50 | 16 | — | |
PRUQRKPURHYKRP
|
7.2 | Ki | 16 | — | |
VAVBWHIBLOPOEM
|
7.2 | Ki | 16 | — | |
IOOGUHXPDYRXFJ
|
7.2 | IC50 | 16 | — | |
WCYJVRQPVHPWLQ
|
7.2 | Ki | 16 | — | |
WHEUGJHMVJCNEP
|
7.2 | IC50 | 16 | — | |
SINAJPKUKOSXOT
|
7.2 | IC50 | 16 | — | |
LPOZDKMXSPAATL
|
7.2 | Ki | 16 | — | |
VOZOMZWSLGQRKP
|
7.1 | IC50 | 16 | — | |
YBRXFNLNMSTVNQ
|
7.1 | IC50 | 16 | — | |
HRTSOMLTEJFUCO
|
7.1 | IC50 | 16 | — | |
PGTVWKLGGCQMBR
|
7.1 | IC50 | 16 | — | |
OMQHFPMEAPEGTA
|
7.1 | Ki | 16 | — | |
AEYRTFCCYIWUJJ
|
7.1 | Ki | 16 | — |