Target Details
UniProt ACP48169
Gene SymbolGABRA4
Protein NameGamma-aminobutyric acid receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 364
  • Clinical molecules 0
  • Avg pChEMBL 7.31
Top Co-occurrence Targets
Active Molecules (364)
InChIKey pChEMBL Type Targets Clinical
ACMQMUZDLQDWTK 8.3 Ki 16
GOCZPCXRIJMRNR 8.3 Ki 16
PHOATQSOBKATTD 8.3 Ki 16
PTRXPVDOTUGGHW 8.3 IC50 16
QWWODAPIEHJFQG 8.3 IC50 16
ZWWZTFYQCITUTK 8.3 IC50 16
BTLWEEGNXUJKKB 8.2 IC50 16
KIVQXKXZISOGBE 8.2 Ki 17
NKIYALPHXLYICR 8.2 IC50 16
YUSWMAULDXZHPY 8.2 Ki 20
ZRRVSALMQDOQAX 8.2 Ki 16
BDISWVKOOATATE 8.2 Ki 16
YUOOYQDBXTWPKL 8.2 Ki 16
OTQXKRRISJPTFS 8.2 IC50 16
WMCJJXHYPNOCMT 8.2 IC50 16
ZRPUPUBWCXFOCY 8.2 Ki 16
NGWYCOVARFKQDW 8.1 Ki 9
DKCAUMRZSZVJCP 8.1 Ki 16
IVGTVZGLPHBTJV 8.1 IC50 16
IVGTVZGLPHBTJV 8.1 IC50 16
QVIQGNJPFOVZBZ 8.1 Ki 16
YHNNMZUUFMJQQY 8.1 IC50 16
XGJLRKVQXMSBJW 8.1 IC50 16
KWPOKTUWXDCATM 8.0 IC50 16
AAOVKJBEBIDNHE 8.0 IC50 16
HQJSGBKPXYZTRN 8.0 IC50 16
MBZNSAJBODIJCK 8.0 IC50 16
HFPZDEHIDKJZSN 8.0 Ki 16
LMJMBPXKXWIKQK 8.0 IC50 16
NNHRCSJWUBQYQV 8.0 IC50 16
PKJGSRHYDOGGLB 8.0 Ki 17
ZJQHPWUVQPJPQT 8.0 IC50 17
FJLMOGVUSSSKEC 7.9 Ki 16
LLAKESJIQFAQJA 7.9 IC50 16
WAPAOOACIDZLKD 7.9 Ki 8
CNVQMRWAJHEFGZ 7.9 Ki 16
OPMIQGMTRGXAQY 7.9 IC50 16
VAARLVBAANTQOM 7.9 Ki 16
HSEWUGOOPIEKBZ 7.9 IC50 16
XAMVDLCXXPEEEG 7.9 Ki 16
YLRURIRIQRAQJJ 7.9 Ki 16
GADIKQPUNWAMEB 7.8 Ki 5
WAEXHEOACCAOSS 7.8 Ki 16
IMMPJABTWMVMPJ 7.8 Ki 16
IQXJMMLNUIUGIQ 7.8 Ki 16
OFBIFZUFASYYRE 7.8 Ki 16
PNRLOCDAUHBIHX 7.8 IC50 16
CKZVPJOTELQSHC 7.8 IC50 16
QCHBQARHFYCDNV 7.8 IC50 16
ZFPVOBQMGRHOBJ 7.8 IC50 16
2D structure