Target Details
UniProt ACP48169
Gene SymbolGABRA4
Protein NameGamma-aminobutyric acid receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 364
  • Clinical molecules 0
  • Avg pChEMBL 7.31
Top Co-occurrence Targets
Active Molecules (364)
InChIKey pChEMBL Type Targets Clinical
MZFKWSFOAVBLQM 9.8 IC50 16
WFPXOWCKXUEKCA 9.7 IC50 16
KVKWRJDNIJTMGN 9.6 IC50 16
QUUNMICPMYIHFS 9.4 IC50 16
XKENJWNGLCKOBP 9.3 IC50 16
NJUMMJUUDUYSKB 9.3 IC50 16
ALBKMJDFBZVHAK 9.3 IC50 16
BYMDBFGHCDTBMT 9.3 IC50 16
IUHKSTINHDUYRO 9.3 IC50 16
VJVAWKPXJCDEQG 9.3 IC50 16
WRXDVVALWQGPMW 9.3 IC50 16
BLJPKQXXDFIIFR 9.2 IC50 16
XJMIBNLJFYSGAR 9.2 IC50 16
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
VZKRZUPJCVFVGR 9.1 IC50 16
DGBIGWXXNGSACT 9.1 Ki 16
QORLMYYHZLDYOR 9.1 Ki 9
YJZGQBGGTBIAOP 9.1 IC50 16
AQKFCEWRKDXGMK 9.0 Ki 16
IPHSQMSRIWZULE 9.0 Ki 16
KDMMIKQMHNBKAV 9.0 Ki 17
RLFKILXOLJVUNF 9.0 IC50 16
BSBLYLUAUVTSMM 9.0 IC50 16
OJLYUGSSUKAWJC 8.8 Ki 16
KVKYGVOAHGNAKZ 8.7 IC50 16
QTEUJQNPMLXVLL 8.7 IC50 16
ZOCSXAVNDGMNBV 8.6 IC50 16
BBSNJCBFCWNPBH 8.6 Ki 8
CHIFCDOIPRCHCF 8.6 IC50 16
CHQPOBHNDRMXFK 8.6 Ki 18
KVKYGVOAHGNAKZ 8.5 IC50 17
LENHHZQGSWCZJW 8.5 Ki 16
NEOUOHDNZDRDNJ 8.5 IC50 16
QIZPCEVRKTWHIE 8.5 IC50 16
RYLDZJANGRBUGW 8.5 IC50 16
MVBVNOZDVRVMNH 8.4 IC50 16
ACUNYYFYYWOKOD 8.4 IC50 16
AXPGZURVLRWNBR 8.4 Ki 16
BZVWONIGXAYZIT 8.4 IC50 16
CDWXZILKRXSANI 8.4 IC50 16
DYSDYZCGZCYPCT 8.4 IC50 16
JTYYMOMTGZSRFM 8.4 IC50 16
LMXUGQJMQSMLIQ 8.4 Ki 17
UFTKNTUWDMJOIX 8.4 IC50 16
UULFOYXSWNADTF 8.4 IC50 16
MKNXZRAKHYWDOS 8.4 IC50 16
XQUJTESAXUTXNH 8.4 Ki 16
YGKSPOBIXHTPMV 8.3 IC50 16
2D structure