Target Details
UniProt ACP48058
Gene SymbolGRIA4
Protein NameGlutamate receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd)
Summary
  • Multi-target molecules 103
  • Clinical molecules 0
  • Avg pChEMBL 6.85
Top Co-occurrence Targets
Active Molecules (103)
InChIKey pChEMBL Type Targets Clinical
DWEFIBGLGPTBOX 6.8 IC50 4
MMCVENIYCFWXTF 6.8 Ki 4
SEVVPWOEIHLQGH 6.7 Ki 4
GQACRJYBZAMVBS 6.7 Ki 4
YUUMCVSQULVXBC 6.7 Ki 3
GCHCBODHULQTMN 6.7 Ki 4
IEBVITXSHAFLJR 6.7 Ki 4
DZZGPRKYOVWBQL 6.7 Ki 4
HYXRLESSUQXLHP 6.6 Ki 4
QLTDMOYTDMCUFF 6.6 Ki 4
JASCMFDYTJFEAR 6.6 IC50 4
CVQAHSMQXIWVLD 6.6 Ki 4
RWVIMCIPOAXUDG 6.5 IC50 11
UCTNZJNATOCSCH 6.5 Ki 4
DBWPFHJYSTVBCZ 6.5 Ki 4
GFBKEXLXXAYEAN 6.5 IC50 4
RPXVIAFEQBNEAX 6.5 IC50 4
IAWXTSMHXFRLQR 6.5 IC50 4
OQCIHSFMLURANM 6.5 IC50 5
FNXUJFFLRGBKLM 6.4 Ki 4
VUYXWDSZUHMHRT 6.4 Ki 4
FTNICLJXPYLDAH 6.4 IC50 3
IYXKOVFPNWKUPM 6.4 IC50 3
JLUIVZIFGHVQKL 6.4 IC50 4
BICPPLXRHOQXDM 6.3 Ki 4
HEHLSRRDKJVHOM 6.3 Ki 4
AEKIJKSVXKWGRJ 6.3 Ki 4
YZSBXDRTJNDPDR 6.3 IC50 4
VTWXNIYVJOMEKC 6.3 Ki 4
DRSBUYJJPSUTFO 6.3 Ki 4
FOOYZANHOGCPSP 6.3 Ki 2
PJQRHOIDKSEWFE 6.3 Ki 2
XTTJVGFNQFHWPI 6.2 IC50 4
QBCVGLJGAYPHNK 6.2 Ki 4
MQFAYNCEKGLLKI 6.2 IC50 4
WXUBLMKEFDTLAG 6.2 Ki 4
NZJUQOAVHJUPHZ 6.2 IC50 4
GEEFQPZFVXQGCJ 6.2 IC50 4
GXLYWXMBTOIUTQ 6.2 IC50 4
KZFIZNJSPIBCFN 6.2 Ki 4
ZPJJGAUEQIVPRW 6.2 IC50 4
LUIPVVRVNKNJEK 6.1 Ki 5
YGSXLTANQIVRPQ 6.1 IC50 4
LBRZSCJIEHCPKW 6.1 Ki 4
OOIMGNLMHOCHOG 6.1 Ki 4
WHUUTDBJXJRKMK 6.1 Ki 5
WHUUTDBJXJRKMK 6.1 Ki 20
IFNJBSHPAUZGBB 6.0 Ki 4
MCKOVZZCGOMMIB 6.0 Ki 6
AXXYLTBQIQBTES 6.0 Ki 4
2D structure