Target Details
UniProt ACP48058
Gene SymbolGRIA4
Protein NameGlutamate receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01094 (ANF_receptor) PF00060 (Lig_chan) PF10613 (Lig_chan-Glu_bd)
Summary
  • Multi-target molecules 103
  • Clinical molecules 0
  • Avg pChEMBL 6.85
Top Co-occurrence Targets
Active Molecules (103)
InChIKey pChEMBL Type Targets Clinical
YXLQKZHKWIKJKC 8.6 Ki 5
UBGQQPPNOYSQQD 8.4 Ki 4
MAEGSWBPNOKENQ 8.4 Ki 4
WYJNVGSFRNBGEH 8.4 Ki 9
YXQUINDTMKETDY 8.4 Ki 9
ONWXFZVXNOZZFR 8.3 Ki 9
PIWNUFICDRESOQ 8.3 Ki 9
QSNIAABEHJATJE 8.2 Ki 4
ZNCDBRBMBIJVRT 8.1 Ki 4
WBDQJMDMOVDHIN 7.8 Ki 4
AEFZZVQZPBFFPN 7.8 Ki 4
HREVLFOANBUFKJ 7.7 Ki 4
ORECTEKXMCPJTB 7.7 Ki 4
PPGDECVBLABBED 7.7 Ki 4
SHDXFFZFHNPBJX 7.7 Ki 4
MLIKVWYGUKDINC 7.7 Ki 4
OFUSRUGBBIJORN 7.7 Ki 4
YXLQKZHKWIKJKC 7.5 IC50 4
UUDAMDVQRQNNHZ 7.4 IC50 5
RKKOVPYSRPVXQY 7.3 Ki 4
RSWNHIRFWDYIOD 7.3 Ki 4
FEIZTUVTFIGEKQ 7.3 Ki 4
FVUZUGGMRGEXCS 7.2 Ki 4
URWGATGVZXHWNI 7.2 Ki 4
GDZVLWJCLHAHHI 7.2 Ki 4
OJHOOLBVWGXREO 7.2 Ki 4
BIUNZQNSKOQDRU 7.2 Ki 4
KTYABWSAGQKAPP 7.2 Ki 9
DBBCCRSHNIGAHB 7.2 Ki 4
GDAQQIJFABGZJS 7.1 Ki 4
XVFDQHLTMSIMNT 7.1 Ki 4
MKDNTSIRYSOGBX 7.1 Ki 4
GDSGJOIKTYTOQG 7.1 IC50 4
UUDAMDVQRQNNHZ 7.1 Ki 4
SNQRPZWKEMQXLW 7.0 Ki 3
QEGZVBVIVYRNHK 7.0 IC50 4
IZRSJUXQYXKNIW 7.0 Ki 4
DTWMIIXDZMYBFK 7.0 Ki 4
UQNAFPHGVPVTAL 6.9 Ki 4
ZUBRKTQZZTVOSA 6.9 IC50 4
GBWIZNYOJITVFI 6.9 Ki 4
DVKDTKVRVXOOED 6.8 IC50 4
IPDQBXQCJNLMHR 6.8 Ki 4
OCEDPPPKQBHDND 6.8 Ki 4
OZXHCFIYEAGHJE 6.8 Ki 4
QYMZRTSHYZACQA 6.8 Ki 4
AEDLNEYZMCRALO 6.8 IC50 4
CLMOKKBBLYYTDT 6.8 IC50 4
JXMKTUJSOCNULB 6.8 Ki 11
WTNVVGMYDRFBPY 6.8 Ki 4
2D structure