Target Details
| UniProt AC | P48048 |
|---|---|
| Gene Symbol | KCNJ1 |
| Protein Name | ATP-sensitive inward rectifier potassium channel 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01007 (IRK) PF17655 (IRK_C) |
Summary
- Multi-target molecules 29
- Clinical molecules 0
- Avg pChEMBL 6.96
KEGG Pathways (2)
Associated Diseases (1)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DBRBZVDPIWOVAV
|
8.7 | Ki | 3 | — | |
NRCYDDLRPFXMNA
|
8.2 | IC50 | 2 | — | |
OCKGFTQIICXDQW
|
8.1 | IC50 | 2 | — | |
COWLYZRDJTYXQV
|
8.0 | IC50 | 2 | — | |
AMJYDFFNPACSTJ
|
7.6 | IC50 | 2 | — | |
OTJQQIAODOJEAU
|
7.3 | IC50 | 2 | — | |
XPHJICKYBJRKLW
|
7.3 | IC50 | 2 | — | |
GKZBQPSXHBJOPU
|
7.3 | IC50 | 2 | — | |
UIGDPUDQDMXRLV
|
7.3 | IC50 | 2 | — | |
SDFXSBFOVNINTE
|
7.1 | IC50 | 2 | — | |
XPWXBGYLYLSHTG
|
7.1 | IC50 | 2 | — | |
LJCOFEDAMMEFHX
|
7.0 | IC50 | 2 | — | |
PLCSPMWUVPYGEZ
|
7.0 | IC50 | 2 | — | |
QIAOITGKSVWAFJ
|
7.0 | IC50 | 2 | — | |
VWVVYFJIUBMXBZ
|
7.0 | IC50 | 2 | — | |
AOWSHKSCOCMIOV
|
6.8 | IC50 | 2 | — | |
YVHUVIOZANOSIW
|
6.8 | IC50 | 2 | — | |
SEWIXNYQXNASBQ
|
6.8 | IC50 | 2 | — | |
SFKBOTCVPFRCEE
|
6.6 | IC50 | 2 | — | |
ITKLWGVJMIJZNQ
|
6.5 | IC50 | 2 | — | |
CIHRMKSTNVZPFD
|
6.5 | IC50 | 2 | — | |
GQOXXKSNEOMYOB
|
6.5 | IC50 | 2 | — | |
AMKWVRGTVQDBBV
|
6.4 | IC50 | 2 | — | |
RWPWIJKKWCFKJJ
|
6.3 | IC50 | 2 | — | |
HXVNLBDKDPCJNH
|
6.3 | IC50 | 2 | — | |
GFZFUQFFPIRNGH
|
6.2 | IC50 | 2 | — | |
UMQXZSKUBTWYIX
|
6.1 | IC50 | 2 | — | |
HXTQUDYQICAAJV
|
6.0 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |