Target Details
| UniProt AC | P48039 |
|---|---|
| Gene Symbol | MTNR1A |
| Protein Name | Melatonin receptor type 1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 916
- Clinical molecules 1
- Avg pChEMBL 8.09
KEGG Pathways (2)
Active Molecules (916)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UROBQRKWWWYDEL
|
10.3 | Ki | 2 | — | |
UTTJOBWIFXQZNV
|
10.3 | Ki | 2 | — | |
VKTMPSYAAVEMEO
|
10.3 | Ki | 2 | — | |
YSLIKCKRXZNCIC
|
10.3 | Ki | 2 | — | |
ZXCZVCUUILSBAR
|
10.3 | Ki | 2 | — | |
UTLRQLQDJLNKNY
|
10.3 | Ki | 2 | — | |
XLQWMAYNSQHNTQ
|
10.3 | Ki | 3 | — | |
FNHLXIXCQDGUCQ
|
10.2 | Ki | 2 | — | |
GBQSWEMPGGYIKG
|
10.2 | Ki | 2 | — | |
OFCLARYYBGKCHN
|
10.2 | Ki | 2 | — | |
QJYZZZMBUAEWOY
|
10.2 | Ki | 2 | — | |
VJGODNYYEUTWJZ
|
10.2 | Ki | 2 | — | |
IZDHETWMKYCGAU
|
10.2 | Ki | 2 | — | |
QKPXFSKGGAUJNY
|
10.2 | IC50 | 2 | — | |
FJDDSMSDZHURBJ
|
10.2 | Ki | 3 | — | |
VPQSZGPHOIJAFK
|
10.2 | IC50 | 2 | — | |
QYFZRIVETVFWFY
|
10.2 | Ki | 2 | — | |
BIDDLRZUESRXIV
|
10.2 | Ki | 2 | — | |
NSEAOKKQWABVSA
|
10.2 | Ki | 2 | — | |
BURWKXUNJOXCGV
|
10.1 | Ki | 3 | — | |
UOVGAGSCHHZUPU
|
10.1 | Ki | 2 | — | |
JDFVYDLICOGWLH
|
10.1 | IC50 | 2 | — | |
HEWLIENXMUSPDG
|
10.1 | IC50 | 2 | — | |
HEWLIENXMUSPDG
|
10.1 | IC50 | 2 | — | |
PCIZTNLLMNKOKT
|
10.1 | Ki | 2 | — | |
RKHCTAKUYDTFHE
|
10.1 | Ki | 2 | — | |
SSMGLPFXFMFFBY
|
10.1 | Ki | 3 | — | |
ZUNXJARMQXSYKS
|
10.1 | Ki | 2 | — | |
FAWBDXMORMETMR
|
10.1 | IC50 | 2 | — | |
GIJVMVBEOMPBKW
|
10.1 | Ki | 2 | — | |
VDBKGGONHKGNTE
|
10.1 | Ki | 2 | — | |
JROBZLKCLLSHNV
|
10.0 | IC50 | 2 | — | |
JWIMNHBXUJNYCZ
|
10.0 | IC50 | 2 | — | |
IYQPCZUAICYGRH
|
10.0 | Ki | 2 | — | |
BCKYGUZOGCRTFP
|
10.0 | Ki | 2 | — | |
CCRUCMHMQXUZAT
|
10.0 | IC50 | 2 | — | |
DLLIXCPIPVUEBH
|
10.0 | Ki | 3 | — | |
DMQVDZBLVXWQQW
|
10.0 | IC50 | 2 | — | |
FZECXOJUPOTGGG
|
10.0 | Ki | 2 | — | |
LBLXNWAPKXWSIO
|
10.0 | Ki | 2 | — | |
OGNIKEZMPYZWPL
|
10.0 | Ki | 2 | — | |
SUFMDDIORSWOHT
|
10.0 | Ki | 2 | — | |
YJYPHIXNFHFHND
|
10.0 | Ki | 5 | — | |
YWDAYXLSFSLOML
|
10.0 | Ki | 2 | — | |
GVOWMRKLYWGZOG
|
9.9 | Ki | 2 | — | |
SDSGISCYQWUIMI
|
9.9 | Ki | 2 | — | |
DUVQUANDZLREPW
|
9.9 | Ki | 2 | — | |
UOVGAGSCHHZUPU
|
9.9 | Ki | 3 | — | |
AUJCIORXQAONNC
|
9.8 | Ki | 2 | — | |
FTZVUKIJZSOGMD
|
9.8 | IC50 | 2 | — |