Target Details
| UniProt AC | P47900 |
|---|---|
| Gene Symbol | P2RY1 |
| Protein Name | P2Y purinoceptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 8
- Clinical molecules 0
- Avg pChEMBL 7.25
KEGG Pathways (5)
Active Molecules (8)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEOSYRMQDNYEEI
|
9.0 | IC50 | 2 | — | |
SGRORDSPRIKCOQ
|
8.5 | IC50 | 2 | — | |
GKKHXSFPYJSHCX
|
7.8 | IC50 | 2 | — | |
WLMZTKAZJUWXCB
|
7.1 | IC50 | 2 | — | |
FUSMULTWGDSXAX
|
6.6 | Ki | 2 | — | |
CCPLITQNIFLYQB
|
6.5 | IC50 | 2 | — | |
ZISKEYVHHKVKHW
|
6.4 | IC50 | 2 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |