Target Details
| UniProt AC | P47898 |
|---|---|
| Gene Symbol | HTR5A |
| Protein Name | 5-hydroxytryptamine receptor 5A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 120
- Clinical molecules 7
- Avg pChEMBL 7.0
KEGG Pathways (4)
Active Molecules (120)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LGSGJWDXMWVXEB
|
6.1 | Ki | 6 | — | |
QBWLTDPVSJCLIE
|
6.0 | Ki | 15 | — | |
CJKGAQSNLYKBKH
|
6.0 | Ki | 9 | — | |
DTJJOPFHDLSVKA
|
6.0 | Ki | 6 | — | |
DZXZPVGWRZCXDH
|
6.0 | Ki | 20 | — | |
HEDOODBJFVUQMS
|
6.0 | Ki | 12 | — | |
ALRBWNXPNRLJKC
|
6.0 | Ki | 10 | — | |
VDHAWDNDOKGFTD
|
6.0 | Ki | 11 | — | |
WEGLOYDTDILXDA
|
6.0 | Ki | 22 | — | |
ASXGJMSKWNBENU
|
6.0 | Ki | 12 | Yes | |
CEUORZQYGODEFX
|
6.0 | Ki | 31 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
MDLAAYDRRZXJIF
|
6.0 | Ki | 22 | — | |
MQLWANLDQKRYQY
|
6.0 | Ki | 8 | — | |
MWRXFEODZOVBTP
|
6.0 | Ki | 3 | — | |
QLOOWOVVZLBYHU
|
6.0 | Ki | 7 | — | |
QZUDBNBUXVUHMW
|
6.0 | Ki | 39 | Yes | |
RAPZEAPATHNIPO
|
6.0 | Ki | 28 | Yes | |
YOGJZQGRTVMCPY
|
6.0 | IC50 | 17 | — | |
ZZZQXCUPAJFVBN
|
6.0 | Ki | 7 | — |