Target Details
UniProt ACP47898
Gene SymbolHTR5A
Protein Name5-hydroxytryptamine receptor 5A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 120
  • Clinical molecules 7
  • Avg pChEMBL 7.0
Top Co-occurrence Targets
Active Molecules (120)
InChIKey pChEMBL Type Targets Clinical
UDUQYNVUNNDSEJ 7.0 Ki 3
JUQLTPCYUFPYKE 7.0 Ki 25
KYIGOCCCBXRHNJ 7.0 IC50 43
LWVFMDTWYOYNOZ 7.0 Ki 3
CWLJQCPGPBYWFX 6.9 Ki 8
ZSENANRQFIMKNZ 6.9 Ki 3
ZSTKHSQDNIGFLM 6.8 Kd 22
BTOJYCTUJJHANF 6.8 Ki 5
AESLFLSZEVKRCB 6.8 Ki 3
OGIMCDMIYGVEHU 6.8 Ki 3
QEGMGDYIJDZJCI 6.8 Ki 10
BQEDZLDNNBDKDS 6.8 Ki 5
QZAYGJVTTNCVMB 6.8 IC50 17
ZKIAIYBUSXZPLP 6.8 Ki 29
ATKUMLMUBZNHEI 6.7 Ki 3
IKBKZGMPCYNSLU 6.7 Ki 13
MLGNCAXDEPBXNR 6.7 Ki 3
YVENIGOVHPMTDH 6.7 Ki 23
GROYHNLGVCIQOI 6.7 Ki 8
YQNWZWMKLDQSAC 6.7 Ki 15
DDIYHVZHGLOJAJ 6.6 Ki 6
GKTQBPYMIGXPKG 6.6 Ki 21 Yes
GKTQBPYMIGXPKG 6.6 Ki 18
QQZUXIPREWBYRJ 6.6 Ki 4
BEQGDXQEYTWVNB 6.6 Ki 7
IKYFNUXRYHSJTJ 6.5 Ki 2
CDTNDXMWHPCPSH 6.5 Ki 6
KIJXVALDJPUIFM 6.5 Ki 6
PKQCAZLGEGUDLP 6.4 Ki 7
BBZITZYOZCKXED 6.4 Ki 8
ODCAEXNEGXTNBY 6.4 Ki 6
UQNXMCNVFPEPNB 6.4 Ki 8
NSASZAUFRUOUIN 6.4 Ki 5
SVJMLYUFVDMUHP 6.4 Ki 26
IQDAWMWSGXPSNV 6.3 Ki 6
KNZNKJDEMHGXSO 6.3 Ki 6
KQKPFRSPSRPDEB 6.3 IC50 9
IAKYDYYOYGXWAX 6.3 Ki 7
MWULMTACIBZPGN 6.2 Ki 8
ZFLRVRLYWHNAEC 6.2 Ki 6
XMHPSFHTLVKATH 6.2 Ki 4
DMULVCHRPCFFGV 6.2 Ki 16
XXJMPUMRHCNWPW 6.2 Ki 8
RGVBFCBKZDWNNA 6.2 Ki 5
UNDVSLNGLPEGMR 6.2 Ki 7
DVSMVUMYJDOPJQ 6.1 Ki 16
MNHDKMDLOJSCGN 6.1 Ki 23
IENZQIKPVFGBNW 6.1 Ki 11 Yes
REJFPXMKRRYBSC 6.1 Ki 3
GXGVWEMSSIKHOZ 6.1 Ki 8
2D structure