Target Details
UniProt ACP47898
Gene SymbolHTR5A
Protein Name5-hydroxytryptamine receptor 5A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 120
  • Clinical molecules 7
  • Avg pChEMBL 7.0
Top Co-occurrence Targets
Active Molecules (120)
InChIKey pChEMBL Type Targets Clinical
OPCCXGXGEHABFP 9.8 Kd 17
CQUWKHKELQQYRI 9.0 IC50 4
CQUWKHKELQQYRI 9.0 IC50 4
BCGWQEUPMDMJNV 9.0 IC50 30 Yes
XFMPGBXLGWZMQP 8.8 Ki 5
KNZNKJDEMHGXSO 8.7 Ki 6
DWIXBLOYUJIYNT 8.7 Ki 6
BKRGVLQUQGGVSM 8.5 Ki 26 Yes
VZZRHPWRULQIJU 8.3 Ki 5
CKSKIWUQLNHIJX 8.3 Ki 6
XFMPGBXLGWZMQP 8.3 Ki 4
KNZNKJDEMHGXSO 8.2 Ki 6
QZNXPVYAMUSJAD 8.2 Ki 5
SCKPQZMXGISHHF 8.2 Ki 5
SEQAMPXQRKYYQF 8.2 Ki 11
NTQGRGIDSHBSJY 8.2 Ki 5
JDPGHZDOBUGUDU 8.2 Ki 5
VAYOSLLFUXYJDT 8.1 Ki 19
CWVMKYZWIKCBIY 8.0 Ki 5
JDPGHZDOBUGUDU 8.0 Ki 4
OVCRQVHRSLIVTD 8.0 Ki 4
DUKNIHFTDAXJON 7.9 Ki 11
DUKNIHFTDAXJON 7.8 Ki 13
DUKNIHFTDAXJON 7.8 Ki 16
DUKNIHFTDAXJON 7.7 Ki 17
XCGSFFUVFURLIX 7.7 Ki 17
WKZLNEWVIAGNAW 7.7 Ki 11
ADOGGHZNEGBRNB 7.7 Ki 4
PZVDYPMNMHJRDU 7.7 Ki 4
JBVXDZODHTVXQZ 7.6 Ki 4
PGMNDAZLZGOWHP 7.6 Ki 5
XIMFQVXENHJKEO 7.6 Ki 10
XIMFQVXENHJKEO 7.6 Ki 10
ZRMFHWUDQQZCJM 7.6 Ki 4
DUKNIHFTDAXJON 7.6 Ki 12
NWEWYDOUXVOLQN 7.5 Ki 4
LUZRJRNZXALNLM 7.5 Ki 20
XHZPPFKLWGSAMV 7.5 Ki 4
VNICFCQJUVFULD 7.4 Ki 15
VBKOTIVQMCTTAQ 7.4 Ki 5
UNRCJLILBVLZDQ 7.3 Ki 6
UNRCJLILBVLZDQ 7.3 Ki 6
HWKROQUZSKPIKQ 7.2 Ki 10
SPCIYGNTAMCTRO 7.2 Ki 15
RKRVRTJVCWZOQS 7.1 Ki 4
MICIQKQOEFSTDP 7.1 Ki 3
BTTOYOKCLDAHHO 7.1 Ki 10
YTYPKXGCVRKLLN 7.0 Ki 5
JZCULFYPORSPJU 7.0 Ki 3
QZPUSPUBLDWGKU 7.0 Ki 3
2D structure