Target Details
| UniProt AC | P47871 |
|---|---|
| Gene Symbol | GCGR |
| Protein Name | Glucagon receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 167
- Clinical molecules 1
- Avg pChEMBL 7.31
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VOSMSHCJSJBJOD
|
6.5 | IC50 | 2 | — | |
NPMZBYQQJWHAEW
|
6.5 | IC50 | 2 | — | |
RFNVDMKXJPQRBI
|
6.4 | IC50 | 2 | — | |
SWIPDZUQVCOFTP
|
6.4 | IC50 | 2 | — | |
YOFQALFMYOUGSF
|
6.4 | IC50 | 2 | — | |
RSJWMKGJEAKNNJ
|
6.4 | Ki | 2 | — | |
CPLKJAOVKQRYLU
|
6.4 | IC50 | 5 | — | |
XFJBPPZDGUTGDU
|
6.3 | IC50 | 2 | — | |
ZPXPEKQMLOAPLT
|
6.3 | IC50 | 15 | — | |
BJXGEYDZUISYLS
|
6.3 | IC50 | 5 | — | |
GFHBMDLZPIDPHI
|
6.3 | IC50 | 2 | — | |
PFOUJNFXNRYXCU
|
6.2 | IC50 | 2 | — | |
MHSKRZAFVKHGJT
|
6.2 | IC50 | 2 | — | |
UEOWVVNOBYAFMV
|
6.1 | IC50 | 2 | — | |
QGUIDVPVMJAYTK
|
6.1 | IC50 | 2 | — | |
IAAZVAITVNPXCO
|
6.1 | IC50 | 5 | — | |
HDUQKBUHXYJBEX
|
6.0 | IC50 | 5 | — |