Target Details
| UniProt AC | P47871 |
|---|---|
| Gene Symbol | GCGR |
| Protein Name | Glucagon receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 167
- Clinical molecules 1
- Avg pChEMBL 7.31
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IOTPUQIURNWCBL
|
7.0 | IC50 | 2 | — | |
VDRBYJICTVBZID
|
7.0 | IC50 | 2 | — | |
WBTZEYLGSORECL
|
7.0 | IC50 | 5 | — | |
BKFPJEBZTCJJRP
|
7.0 | IC50 | 2 | — | |
MYFXPJIUHYQWRX
|
7.0 | IC50 | 2 | — | |
DRBYFBHVRFFBIU
|
7.0 | IC50 | 2 | — | |
JYBVCXGFJLXTCP
|
7.0 | Ki | 2 | — | |
MDDANNKYTHKAHR
|
7.0 | IC50 | 2 | — | |
UPYHVTCMTMZKAX
|
7.0 | IC50 | 12 | — | |
XBOAMGVRMOKHNU
|
7.0 | IC50 | 6 | — | |
BEUJQOCLEVYLAY
|
7.0 | IC50 | 5 | — | |
DKZILDKFHNFIHZ
|
7.0 | IC50 | 2 | — | |
NBCXZLPCCIVOKY
|
7.0 | IC50 | 5 | — | |
WPHHXNCBGPKNOY
|
6.9 | IC50 | 2 | — | |
KZLCRRAGBNSUBK
|
6.9 | IC50 | 5 | — | |
MYYKZRMEYNXGOG
|
6.9 | IC50 | 2 | — | |
NGUABMKOSJANPJ
|
6.9 | IC50 | 2 | — | |
AZBHFSLUTGHEPH
|
6.9 | IC50 | 6 | — | |
SLYYRVVPLWMNPO
|
6.9 | IC50 | 2 | — | |
FDAPJZJLEIYQAN
|
6.9 | IC50 | 2 | — | |
GSQDVEYSGMKGJU
|
6.9 | IC50 | 2 | — | |
CHYPABFSTPTACZ
|
6.8 | IC50 | 2 | — | |
JTMDOZVHCVTETN
|
6.8 | IC50 | 2 | — | |
SLEDJBMFRMKJLH
|
6.8 | IC50 | 5 | — | |
RRGXAHXPWSPEEU
|
6.8 | IC50 | 2 | — | |
OLORAIPIPRFIOH
|
6.8 | IC50 | 2 | — | |
QUKMNFBZSMFVFB
|
6.8 | IC50 | 5 | — | |
BYRKVDOSQUAVAB
|
6.8 | IC50 | 5 | — | |
KVOWJSITTRQRSW
|
6.7 | IC50 | 2 | — | |
PLROHMUOLNMPBX
|
6.7 | IC50 | 2 | — | |
QXROCLPRKWUYBA
|
6.7 | IC50 | 5 | — | |
RYBDMKKIZXATSX
|
6.7 | IC50 | 5 | — | |
XUJSRSRKGLTVPA
|
6.7 | IC50 | 2 | — | |
RCRLRZAUQKXAAX
|
6.7 | Ki | 2 | — | |
FVWMKILDWMMUDG
|
6.7 | IC50 | 2 | — | |
NCECUPUQFBKLMA
|
6.7 | IC50 | 5 | — | |
UTJPXFUHWFHNCZ
|
6.7 | IC50 | 6 | — | |
VNQSYWZBMNSLRL
|
6.7 | IC50 | 2 | — | |
NPMZBYQQJWHAEW
|
6.7 | IC50 | 2 | — | |
QCXYVMFKAJYFNH
|
6.7 | IC50 | 2 | — | |
SZXJKSQEKRRTMT
|
6.6 | IC50 | 5 | — | |
WABICJZHMMDLSC
|
6.6 | Ki | 2 | — | |
FNTGKGUQJOVZES
|
6.5 | Ki | 2 | — | |
GUZODAKISVJZOY
|
6.5 | IC50 | 6 | — | |
IVQRDNQHHJAUCS
|
6.5 | IC50 | 5 | — | |
XKENBIHIHWFSFY
|
6.5 | IC50 | 2 | — | |
ZIRPNTIMTLOHIL
|
6.5 | IC50 | 2 | — | |
VRSHGZMFXJHCDY
|
6.5 | IC50 | 5 | — | |
MDQQAIUZIATVCK
|
6.5 | IC50 | 5 | — | |
QSUCCHXYMZTHEG
|
6.5 | IC50 | 2 | — |