Target Details
| UniProt AC | P47871 |
|---|---|
| Gene Symbol | GCGR |
| Protein Name | Glucagon receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 167
- Clinical molecules 1
- Avg pChEMBL 7.31
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SQCUILFEAKKVAC
|
7.7 | IC50 | 2 | — | |
VHURVYZHODPCCB
|
7.7 | IC50 | 2 | — | |
XNSJRSAITGCUKS
|
7.7 | IC50 | 2 | — | |
KOCYTHSBSWIFSD
|
7.7 | IC50 | 5 | — | |
BZXMLCVDKDXRQY
|
7.6 | IC50 | 2 | — | |
ZGRAABYQGYPWLS
|
7.6 | IC50 | 2 | — | |
VLGOFRLXSHLEAO
|
7.6 | IC50 | 2 | — | |
AUEUQGHVNOSGSL
|
7.5 | Ki | 10 | — | |
DAUDLQFCWWLQPT
|
7.5 | IC50 | 2 | — | |
YXRLENJRMMVUDH
|
7.5 | IC50 | 2 | — | |
COXXCKLSWHHFDS
|
7.5 | IC50 | 5 | — | |
VEXHFZLCFRSPSZ
|
7.5 | IC50 | 2 | — | |
KNMAVSXEMFMOGI
|
7.5 | IC50 | 2 | — | |
XKURAAGCCZEBHF
|
7.5 | IC50 | 2 | — | |
OUZOYODGROMRMW
|
7.4 | IC50 | 2 | — | |
CDMGBJANTYXAIV
|
7.4 | IC50 | 34 | Yes | |
JJGVEWLQTOEULJ
|
7.4 | IC50 | 2 | — | |
KWBJZWKTXONOQI
|
7.4 | IC50 | 5 | — | |
PZQZQDIIWVHESQ
|
7.4 | IC50 | 2 | — | |
KNMAVSXEMFMOGI
|
7.3 | IC50 | 2 | — | |
BOPMXYXKSFCVIW
|
7.3 | IC50 | 2 | — | |
UOXBWPOEKZEVKV
|
7.3 | IC50 | 2 | — | |
MTBJTQZAQADZQL
|
7.3 | IC50 | 2 | — | |
APKKXGAJMPHCEP
|
7.3 | IC50 | 5 | — | |
SVLDQMHFIWDPJO
|
7.3 | IC50 | 2 | — | |
XNNDVZWCQPPMHC
|
7.3 | Ki | 10 | — | |
XNSJRSAITGCUKS
|
7.3 | IC50 | 2 | — | |
JHYVBNOMIUNRJS
|
7.3 | Ki | 2 | — | |
CIDYLAWHEXYTGX
|
7.3 | IC50 | 2 | — | |
FVDONABKZHMTCY
|
7.3 | IC50 | 2 | — | |
BZXMLCVDKDXRQY
|
7.2 | IC50 | 11 | — | |
WGMDTVFTELHPOL
|
7.2 | IC50 | 2 | — | |
AWHRFPLTQPNOTD
|
7.2 | IC50 | 5 | — | |
CWDASHXSVSFWKM
|
7.2 | Ki | 10 | — | |
KVIYSVXFZOEINO
|
7.2 | IC50 | 6 | — | |
KOVJJWYJLGKJAI
|
7.1 | IC50 | 2 | — | |
XTOBAVZIBVVXLS
|
7.1 | IC50 | 2 | — | |
GKFODRKFKVOWTH
|
7.1 | IC50 | 2 | — | |
SGTLXOZGCVZYAN
|
7.1 | IC50 | 2 | — | |
HHLCSKJKCZOHTH
|
7.1 | IC50 | 2 | — | |
QHKYPYXTTXKZST
|
7.1 | IC50 | 28 | — | |
CTOLIBJXQJXWDY
|
7.1 | IC50 | 2 | — | |
OIQWAEIGTZYWRX
|
7.1 | IC50 | 2 | — | |
XEECUIDWJQYSIO
|
7.1 | IC50 | 2 | — | |
FTBIQPJNXCTJIU
|
7.1 | IC50 | 2 | — | |
NVWTWHYQHRAFNN
|
7.1 | IC50 | 2 | — | |
WFUXVTIXEWVFED
|
7.1 | IC50 | 2 | — | |
YZUIGWQMHIUXNA
|
7.1 | IC50 | 2 | — | |
COVWDRBCMJOSQM
|
7.0 | IC50 | 5 | — | |
CTJDFSIKSQVUTF
|
7.0 | IC50 | 2 | — |