Target Details
| UniProt AC | P47871 |
|---|---|
| Gene Symbol | GCGR |
| Protein Name | Glucagon receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 167
- Clinical molecules 1
- Avg pChEMBL 7.31
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (167)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVSVLRYVPXFJOT
|
9.4 | IC50 | 3 | — | |
HNTXQDRFWJBZGO
|
8.6 | IC50 | 2 | — | |
YQWKQQFUAPWMJC
|
8.6 | IC50 | 2 | — | |
CWPADRJBQLPUCB
|
8.6 | IC50 | 3 | — | |
PADIVHKPYLHTDY
|
8.5 | Ki | 10 | — | |
GQPPIAAXSZCKMB
|
8.4 | Ki | 10 | — | |
MRJZJRLNCMMRCZ
|
8.4 | IC50 | 2 | — | |
ZAVYYYQORHVVFN
|
8.4 | IC50 | 4 | — | |
WCVRCGUPWLUXJR
|
8.4 | IC50 | 2 | — | |
UECFQNMLGNHNSO
|
8.3 | IC50 | 2 | — | |
UECFQNMLGNHNSO
|
8.3 | IC50 | 2 | — | |
MYHQPEVOOWDUDW
|
8.3 | IC50 | 2 | — | |
IADKHNLYTDEPGD
|
8.3 | IC50 | 6 | — | |
LOKUGNIDKBRXJC
|
8.3 | IC50 | 2 | — | |
LOKUGNIDKBRXJC
|
8.3 | IC50 | 2 | — | |
QLCNDVIJFAHAFO
|
8.3 | IC50 | 2 | — | |
YDXHIJKYXAXQTE
|
8.2 | Ki | 2 | — | |
KNTOEHKTBLUGLN
|
8.2 | IC50 | 2 | — | |
DCXARCKEWAQLJB
|
8.2 | Ki | 10 | — | |
KHJHACWGMCPAEX
|
8.2 | Ki | 10 | — | |
REIGIHUHXDNPSA
|
8.2 | IC50 | 2 | — | |
SPYNVKYBDKGKEH
|
8.2 | IC50 | 2 | — | |
YFBXBYGXHKOXOG
|
8.2 | Ki | 10 | — | |
UXPYCHMVTKGDJP
|
8.2 | IC50 | 2 | — | |
OBRBSPYTOYTECA
|
8.2 | IC50 | 2 | — | |
HHKKVYXTKFAECF
|
8.1 | IC50 | 2 | — | |
OIQWAEIGTZYWRX
|
8.1 | IC50 | 2 | — | |
QJEGIIJPDLHOEZ
|
8.1 | IC50 | 2 | — | |
ANMUHQCUTMTNRH
|
8.1 | IC50 | 2 | — | |
FPOPGDWXBFUBKQ
|
8.1 | Ki | 10 | — | |
KOZDDXIYVDHLIC
|
8.1 | IC50 | 2 | — | |
SYWXLIGCTNVJDM
|
8.1 | IC50 | 2 | — | |
VERXBCYVZFLZNT
|
8.1 | Ki | 2 | — | |
ICARRUHVPUOWDW
|
8.0 | IC50 | 2 | — | |
OLGWNKHCHXVJMX
|
8.0 | IC50 | 2 | — | |
JTIOTPJAIFIFFX
|
8.0 | Ki | 10 | — | |
OIKPHPKYVGTXMU
|
8.0 | Ki | 10 | — | |
VSGDYFXFEPKTGU
|
7.9 | IC50 | 2 | — | |
ZBMZGBGZOQFXEP
|
7.9 | Ki | 3 | — | |
OTDAFCWROVFKOL
|
7.9 | IC50 | 2 | — | |
OTDAFCWROVFKOL
|
7.9 | IC50 | 2 | — | |
QMZREIRRGCJPTH
|
7.9 | IC50 | 2 | — | |
YDAXDTSMRRYDQR
|
7.9 | IC50 | 2 | — | |
ITDOIINIFNQSFX
|
7.9 | IC50 | 2 | — | |
JKDNPQJPEAQBPC
|
7.8 | IC50 | 2 | — | |
XNSJRSAITGCUKS
|
7.8 | IC50 | 2 | — | |
YAJKYUVXRYCKPC
|
7.8 | IC50 | 2 | — | |
YZUWLDZGWNDIRB
|
7.8 | Ki | 2 | — | |
GLTBMLMTGHGENX
|
7.8 | IC50 | 2 | — | |
AKFRCBAYXPRXSG
|
7.7 | IC50 | 2 | — |