Target Details
| UniProt AC | P47870 |
|---|---|
| Gene Symbol | GABRB2 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 445
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OMGOVFIKWLKTPS
|
6.2 | Ki | 16 | — | |
BZIBRALMCDHACX
|
6.2 | Ki | 17 | — | |
CVZWKJSPJYNXCC
|
6.2 | Ki | 3 | — | |
JWTQJUQJIRWZLA
|
6.2 | Ki | 16 | — | |
ODWCGGCCGLKRAK
|
6.2 | Ki | 16 | — | |
TXPKEBVGMYWHJR
|
6.2 | IC50 | 3 | — | |
ICRYUJPBYIPXQF
|
6.2 | IC50 | 16 | — | |
ZMKDYQONTIIETL
|
6.2 | Ki | 16 | — | |
OJOTYQLMNVPQBO
|
6.2 | Ki | 16 | — | |
RRAXPPHKWFOGGL
|
6.2 | Ki | 16 | — | |
WQIWYEISPHMPOA
|
6.2 | IC50 | 16 | — | |
ARCJBXYEOMXBSZ
|
6.2 | IC50 | 16 | — | |
CTPREUOHTKHCHT
|
6.2 | IC50 | 16 | — | |
DPISUGVHZBSEIR
|
6.2 | IC50 | 3 | — | |
XFUAEWGHLXLENC
|
6.2 | IC50 | 16 | — | |
BSEVRQDRIQMBCV
|
6.2 | IC50 | 16 | — | |
DHEXTYZLLGWEFS
|
6.2 | Ki | 16 | — | |
HBOSSQBJUBOEJN
|
6.1 | Ki | 16 | — | |
IADROWGKULIMIX
|
6.1 | Ki | 3 | — | |
XVFJUDUNNHPHLN
|
6.1 | IC50 | 16 | — | |
HYJUIJYNZHZBOK
|
6.1 | IC50 | 16 | — | |
WJEPRNMCEBRSDB
|
6.1 | IC50 | 16 | — | |
OXSWCVXEQZIBGE
|
6.1 | IC50 | 3 | — | |
YLZBNNDOEUIHFB
|
6.1 | IC50 | 16 | — | |
APPBGPRMFVUPRH
|
6.1 | IC50 | 3 | — | |
CXNUOOTVTMVRCI
|
6.1 | IC50 | 3 | — | |
LKUSWPRPRBXYPH
|
6.1 | IC50 | 16 | — | |
VKMJGKFQKLVODR
|
6.1 | IC50 | 16 | — | |
VAEZVMCCCWEXEH
|
6.1 | Ki | 16 | — | |
ZXYMHGABHZSFOI
|
6.1 | Ki | 16 | — | |
DOOGDICMBOTQOZ
|
6.1 | IC50 | 16 | — | |
KGNWRICPWILABJ
|
6.1 | Ki | 6 | — | |
PJMYDDGWVUCELC
|
6.0 | Ki | 6 | — | |
SLNCMJYPLFSUGO
|
6.0 | Ki | 16 | — | |
SZHSENNQOQSFEA
|
6.0 | IC50 | 16 | — | |
UNBQMUNNSLPLLQ
|
6.0 | Ki | 4 | — | |
DHLJRIFIBJGWBS
|
6.0 | IC50 | 16 | — | |
DQDLJDCSJFQOHI
|
6.0 | IC50 | 16 | — | |
FUULVCWWUPGUMY
|
6.0 | IC50 | 16 | — | |
GCTOZKWOFVUEAW
|
6.0 | IC50 | 16 | — | |
IHFBPDAQLQOCBX
|
6.0 | Ki | 18 | — | |
KVZVPZYFPDOIMI
|
6.0 | IC50 | 16 | — | |
MAVYALTWHWZSCK
|
6.0 | IC50 | 3 | — | |
RYFIWEJRWHTFBM
|
6.0 | IC50 | 16 | — | |
XORHKQBNMFEJKZ
|
6.0 | Ki | 3 | — |