Target Details
| UniProt AC | P47870 |
|---|---|
| Gene Symbol | GABRB2 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 445
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WNDIDYSCZWXEJF
|
6.6 | Ki | 16 | — | |
LOBNIVNGRUTMOS
|
6.5 | IC50 | 16 | — | |
WRUTXEAYYQYJHO
|
6.5 | Ki | 16 | — | |
HJGRBNHROFTASJ
|
6.5 | IC50 | 16 | — | |
QCDKBYHARZQRIV
|
6.5 | Ki | 5 | — | |
YHZXFRGWTKYPKS
|
6.5 | Ki | 16 | — | |
GAQCKHAXURZXGX
|
6.5 | IC50 | 16 | — | |
VEWLYIAEUXDQBW
|
6.5 | IC50 | 16 | — | |
GDVGLPNNOCDLLD
|
6.5 | IC50 | 16 | — | |
UXBYKUXVPASURW
|
6.5 | Ki | 4 | — | |
GEFDSAOHFGLQEZ
|
6.5 | Ki | 17 | — | |
WCTCMHZWHMFZFN
|
6.5 | Ki | 17 | — | |
DDSULWHSYUPHBK
|
6.5 | IC50 | 16 | — | |
XRWYYMUIIXMQBL
|
6.5 | IC50 | 16 | — | |
CVZIRDLTVVTXNF
|
6.4 | Ki | 6 | — | |
DAYQXLQRTQODQF
|
6.4 | Ki | 16 | — | |
DNCFKDLZZSXXJP
|
6.4 | IC50 | 16 | — | |
HOPCRSLMIVRJDL
|
6.4 | Ki | 3 | — | |
RACLCHHASISYPU
|
6.4 | Ki | 4 | — | |
MUPIUJYENVWEKT
|
6.4 | IC50 | 16 | — | |
NQFQEBQBZXSXIX
|
6.4 | IC50 | 16 | — | |
RBMPSWHARBABOC
|
6.4 | Ki | 6 | — | |
VNFZCRPFALLSNM
|
6.4 | IC50 | 16 | — | |
SQPWTARSPNZNEI
|
6.4 | IC50 | 16 | — | |
ZAFYATHCZYHLPB
|
6.4 | Ki | 7 | — | |
DCGKLGYFWMHNPR
|
6.4 | IC50 | 4 | — | |
QCSFXCHHKYXLHE
|
6.4 | Ki | 16 | — | |
YFEZLTPSCJWVHI
|
6.4 | Ki | 16 | — | |
YOJAHANNNITYMX
|
6.4 | Ki | 16 | — | |
ZLAPTIDQRXJQQL
|
6.4 | IC50 | 16 | — | |
RXJAQIBDEJFUCL
|
6.4 | Ki | 6 | — | |
AEPFXRGRJZMVIF
|
6.3 | Ki | 17 | — | |
BHJKLRZKDBSSKN
|
6.3 | Ki | 6 | — | |
JBTLCAMUYYCXTA
|
6.3 | IC50 | 16 | — | |
DKCNNHVHQYMVTO
|
6.3 | IC50 | 16 | — | |
SWLVOEWTHNCIDF
|
6.3 | Ki | 3 | — | |
HMRRNXHWVOACEA
|
6.3 | IC50 | 3 | — | |
BDGWCPYUERFMMY
|
6.3 | Ki | 16 | — | |
UMYWGMKUCZAQJO
|
6.3 | Ki | 16 | — | |
FNZFELZOBRBQJY
|
6.3 | IC50 | 16 | — | |
IGCSLIVTBUKKRS
|
6.3 | IC50 | 16 | — | |
SRJOCJYGOFTFLH
|
6.3 | Ki | 16 | — | |
VFWOXQNFPHOBLO
|
6.3 | IC50 | 3 | — | |
GAGMZQZBWNYDQU
|
6.3 | Ki | 6 | — | |
IKDYRDIWKFJQTR
|
6.3 | IC50 | 16 | — | |
FRKWUXZCSLOPIC
|
6.3 | IC50 | 7 | — | |
PZWMQJZDDYQYGN
|
6.3 | Ki | 16 | — | |
YDLSCFILSJHEPL
|
6.3 | IC50 | 3 | — | |
ZEEOGWVZWOURAE
|
6.2 | Ki | 16 | — | |
NDRWXFUZQPBELD
|
6.2 | IC50 | 3 | — |