Target Details
| UniProt AC | P47870 |
|---|---|
| Gene Symbol | GABRB2 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 445
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZFPVOBQMGRHOBJ
|
7.8 | IC50 | 16 | — | |
PSDFROGPPFTBND
|
7.8 | Ki | 7 | — | |
JWZNKJCEYMWLHS
|
7.8 | IC50 | 16 | — | |
MEWGBPFYMUBENF
|
7.8 | IC50 | 16 | — | |
NAXZRUMPHRMRDF
|
7.8 | IC50 | 16 | — | |
VXOXRIDQOBACKW
|
7.8 | Ki | 16 | — | |
PTTQXDBPTFOCMT
|
7.8 | Ki | 6 | — | |
YJYRFBZSNPRHKU
|
7.8 | IC50 | 16 | — | |
PFSCOMOMUBXDBR
|
7.7 | Ki | 4 | — | |
QVBUOPGWPXUAHT
|
7.7 | IC50 | 16 | — | |
UIPGLQFPZVUUQW
|
7.7 | Ki | 16 | — | |
VQENDYBPFSSMNH
|
7.7 | IC50 | 16 | — | |
BYEKIJACVDAPTD
|
7.7 | Ki | 16 | — | |
LLAKESJIQFAQJA
|
7.7 | IC50 | 16 | — | |
FQDQLHDSVITISC
|
7.7 | IC50 | 16 | — | |
HKLYPSSDHPAOJM
|
7.7 | IC50 | 16 | — | |
RSEMKXACIMVTQP
|
7.7 | Ki | 16 | — | |
WRDHNUVAWMYMJK
|
7.7 | IC50 | 16 | — | |
AURFZBICLPNKBZ
|
7.7 | IC50 | 16 | — | |
YTUMMZANIYQNOM
|
7.7 | Ki | 8 | — | |
ZFLBRINMIQTFNB
|
7.7 | Ki | 18 | — | |
CJYPUCKDMBCYEH
|
7.6 | IC50 | 16 | — | |
GSQMITXEUGIGFD
|
7.6 | Ki | 3 | — | |
LNPSYDJGQQETLB
|
7.6 | Ki | 16 | — | |
SHTOUNSWZVCSOU
|
7.6 | IC50 | 16 | — | |
TWQDMCPDTPVCQP
|
7.6 | IC50 | 16 | — | |
VHQCVUYEMJHQEX
|
7.6 | Ki | 16 | — | |
JHDNCJGODWCHES
|
7.6 | IC50 | 16 | — | |
LIXHLXZPUZQKCT
|
7.6 | IC50 | 16 | — | |
MBBOXTKOOFAZLI
|
7.6 | IC50 | 16 | — | |
PDOZRVXKPBQAJH
|
7.6 | IC50 | 16 | — | |
UHEYIOPHTBWBQN
|
7.6 | IC50 | 3 | — | |
ULDBOWIRGDMZPF
|
7.6 | Ki | 8 | — | |
JWLCOGXPTWMMDY
|
7.6 | Ki | 16 | — | |
KBVJZOBCOIANOX
|
7.6 | Ki | 16 | — | |
KOMBGWPXIHBMLL
|
7.6 | IC50 | 16 | — | |
OSHQANHMWJQRHB
|
7.6 | Ki | 16 | — | |
ULMKSNRBNFFOJQ
|
7.6 | Ki | 16 | — | |
ZWJGDMSWCKASII
|
7.6 | IC50 | 16 | — | |
YMFJMRVJWVJJAB
|
7.6 | Ki | 5 | — | |
HCJVWLPVQMYLOI
|
7.6 | Ki | 8 | — | |
HSUCRXNJMPDNOG
|
7.6 | IC50 | 16 | — | |
IVZIOBTVAJBBAS
|
7.6 | Ki | 5 | — | |
JNWDOTPNEZYWGO
|
7.6 | Ki | 16 | — | |
JAFQEKAQGSQGTM
|
7.6 | Ki | 16 | — | |
KQTMWRZAVOUNCI
|
7.6 | IC50 | 16 | — | |
VIEKPLVJCPXIIB
|
7.6 | IC50 | 16 | — | |
WDTNKNNGHGOKBH
|
7.6 | Ki | 9 | — | |
XLKKKDPUVUIHEL
|
7.6 | IC50 | 16 | — | |
YDLSCFILSJHEPL
|
7.5 | IC50 | 3 | — |