Target Details
| UniProt AC | P47870 |
|---|---|
| Gene Symbol | GABRB2 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 445
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZRRVSALMQDOQAX
|
8.2 | Ki | 16 | — | |
BDISWVKOOATATE
|
8.2 | Ki | 16 | — | |
BGRWSFIQQPVEML
|
8.2 | Ki | 6 | — | |
YUOOYQDBXTWPKL
|
8.2 | Ki | 16 | — | |
OTQXKRRISJPTFS
|
8.2 | IC50 | 16 | — | |
VPZOLJKOURRVNO
|
8.2 | IC50 | 3 | — | |
WMCJJXHYPNOCMT
|
8.2 | IC50 | 16 | — | |
ZRPUPUBWCXFOCY
|
8.2 | Ki | 16 | — | |
OWTXLWRGHNAFHX
|
8.1 | Ki | 6 | — | |
DKCAUMRZSZVJCP
|
8.1 | Ki | 16 | — | |
IVGTVZGLPHBTJV
|
8.1 | IC50 | 16 | — | |
IVGTVZGLPHBTJV
|
8.1 | IC50 | 16 | — | |
QVIQGNJPFOVZBZ
|
8.1 | Ki | 16 | — | |
YHNNMZUUFMJQQY
|
8.1 | IC50 | 16 | — | |
PPLHNABOBXLAJU
|
8.1 | Ki | 4 | — | |
XGJLRKVQXMSBJW
|
8.1 | IC50 | 16 | — | |
QORLMYYHZLDYOR
|
8.0 | Ki | 9 | — | |
FLEQTIDRWGGTRR
|
8.0 | Ki | 7 | — | |
KWPOKTUWXDCATM
|
8.0 | IC50 | 16 | — | |
HQJSGBKPXYZTRN
|
8.0 | IC50 | 16 | — | |
IXGIOXIKQZCZIK
|
8.0 | Ki | 8 | — | |
MBZNSAJBODIJCK
|
8.0 | IC50 | 16 | — | |
PWFUHHSGSJDKCU
|
8.0 | IC50 | 16 | — | |
DVKHCFDZNVGRQT
|
8.0 | IC50 | 16 | — | |
HFPZDEHIDKJZSN
|
8.0 | Ki | 16 | — | |
LMJMBPXKXWIKQK
|
8.0 | IC50 | 16 | — | |
NNHRCSJWUBQYQV
|
8.0 | IC50 | 16 | — | |
PKJGSRHYDOGGLB
|
8.0 | Ki | 17 | — | |
PTJXEJYDOYCHOL
|
8.0 | IC50 | 3 | — | |
UBZGCHSBAOJHLE
|
8.0 | Ki | 3 | — | |
ZJQHPWUVQPJPQT
|
8.0 | IC50 | 17 | — | |
FJLMOGVUSSSKEC
|
7.9 | Ki | 16 | — | |
LLAKESJIQFAQJA
|
7.9 | IC50 | 16 | — | |
AAOVKJBEBIDNHE
|
7.9 | Ki | 16 | — | |
BIBRQTYVULTGSH
|
7.9 | Ki | 4 | — | |
CNVQMRWAJHEFGZ
|
7.9 | Ki | 16 | — | |
OPMIQGMTRGXAQY
|
7.9 | IC50 | 16 | — | |
VAARLVBAANTQOM
|
7.9 | Ki | 16 | — | |
GAONFNHSQRTFJA
|
7.9 | Ki | 6 | — | |
HSEWUGOOPIEKBZ
|
7.9 | IC50 | 16 | — | |
XAMVDLCXXPEEEG
|
7.9 | Ki | 16 | — | |
YLRURIRIQRAQJJ
|
7.9 | Ki | 16 | — | |
OWTXLWRGHNAFHX
|
7.8 | Ki | 6 | — | |
RBMPSWHARBABOC
|
7.8 | Ki | 6 | — | |
WAEXHEOACCAOSS
|
7.8 | Ki | 16 | — | |
IMMPJABTWMVMPJ
|
7.8 | Ki | 16 | — | |
IQXJMMLNUIUGIQ
|
7.8 | Ki | 16 | — | |
PNRLOCDAUHBIHX
|
7.8 | IC50 | 16 | — | |
CKZVPJOTELQSHC
|
7.8 | IC50 | 16 | — | |
QCHBQARHFYCDNV
|
7.8 | IC50 | 16 | — |