Target Details
| UniProt AC | P47870 |
|---|---|
| Gene Symbol | GABRB2 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 445
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OJLYUGSSUKAWJC
|
8.8 | Ki | 16 | — | |
KVKYGVOAHGNAKZ
|
8.7 | IC50 | 16 | — | |
IRYAGFJMRZLHGE
|
8.7 | Ki | 6 | — | |
GTOBFJHFOZIFFU
|
8.7 | Ki | 5 | — | |
QTEUJQNPMLXVLL
|
8.7 | IC50 | 16 | — | |
UKHFPVCOXBJPIN
|
8.7 | IC50 | 17 | — | |
OFBIFZUFASYYRE
|
8.6 | Ki | 16 | — | |
ZOCSXAVNDGMNBV
|
8.6 | IC50 | 16 | — | |
PCKMQUISQMUBKK
|
8.6 | Ki | 4 | — | |
LOZNAQDBHKVLRN
|
8.6 | Ki | 6 | — | |
PPTYJKAXVCCBDU
|
8.6 | Ki | 7 | — | |
OKOKWNYOLUGIGN
|
8.6 | Ki | 3 | — | |
CHIFCDOIPRCHCF
|
8.6 | IC50 | 16 | — | |
CHQPOBHNDRMXFK
|
8.6 | Ki | 18 | — | |
KVKYGVOAHGNAKZ
|
8.5 | IC50 | 17 | — | |
LENHHZQGSWCZJW
|
8.5 | Ki | 16 | — | |
LPAODQAWVMEXKR
|
8.5 | IC50 | 16 | — | |
LZTHAJBUMOQDLU
|
8.5 | IC50 | 3 | — | |
NEOUOHDNZDRDNJ
|
8.5 | IC50 | 16 | — | |
QIZPCEVRKTWHIE
|
8.5 | IC50 | 16 | — | |
RYLDZJANGRBUGW
|
8.5 | IC50 | 16 | — | |
VMKZXEMKFBINKN
|
8.5 | Ki | 3 | — | |
MVBVNOZDVRVMNH
|
8.4 | IC50 | 16 | — | |
ACUNYYFYYWOKOD
|
8.4 | IC50 | 16 | — | |
AXPGZURVLRWNBR
|
8.4 | Ki | 16 | — | |
BZVWONIGXAYZIT
|
8.4 | IC50 | 16 | — | |
CDWXZILKRXSANI
|
8.4 | IC50 | 16 | — | |
DYSDYZCGZCYPCT
|
8.4 | IC50 | 16 | — | |
JTYYMOMTGZSRFM
|
8.4 | IC50 | 16 | — | |
LMXUGQJMQSMLIQ
|
8.4 | Ki | 17 | — | |
UFTKNTUWDMJOIX
|
8.4 | IC50 | 16 | — | |
UULFOYXSWNADTF
|
8.4 | IC50 | 16 | — | |
MKNXZRAKHYWDOS
|
8.4 | IC50 | 16 | — | |
XQUJTESAXUTXNH
|
8.4 | Ki | 16 | — | |
YGKSPOBIXHTPMV
|
8.3 | IC50 | 16 | — | |
ACMQMUZDLQDWTK
|
8.3 | Ki | 16 | — | |
GOCZPCXRIJMRNR
|
8.3 | Ki | 16 | — | |
PHOATQSOBKATTD
|
8.3 | Ki | 16 | — | |
PTRXPVDOTUGGHW
|
8.3 | IC50 | 16 | — | |
QWWODAPIEHJFQG
|
8.3 | IC50 | 16 | — | |
XRRMKGIMNWBQJX
|
8.3 | Ki | 3 | — | |
LJRIFLWERUHAIZ
|
8.3 | Ki | 8 | — | |
ZWWZTFYQCITUTK
|
8.3 | IC50 | 16 | — | |
ZGEGOFCLSWVVKG
|
8.2 | Ki | 5 | — | |
ZFOFJXFVCJQXBL
|
8.2 | Ki | 3 | — | |
BTLWEEGNXUJKKB
|
8.2 | IC50 | 16 | — | |
KIVQXKXZISOGBE
|
8.2 | Ki | 17 | — | |
LIFDPEORUVTOCP
|
8.2 | IC50 | 4 | — | |
NKIYALPHXLYICR
|
8.2 | IC50 | 16 | — | |
YUSWMAULDXZHPY
|
8.2 | Ki | 20 | — |