Target Details
| UniProt AC | P47870 |
|---|---|
| Gene Symbol | GABRB2 |
| Protein Name | Gamma-aminobutyric acid receptor subunit beta-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 445
- Clinical molecules 0
- Avg pChEMBL 7.45
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CGMJQQJSWIRRRL
|
10.1 | Ki | 6 | — | |
LTRYPGNCHZSXSI
|
9.9 | Ki | 3 | — | |
NAGYYVWENUNCDU
|
9.9 | Ki | 3 | — | |
TUYGGVAJDAZCIC
|
9.9 | Ki | 3 | — | |
KKXPFXBGMGQSMA
|
9.8 | Ki | 3 | — | |
MZFKWSFOAVBLQM
|
9.8 | IC50 | 16 | — | |
WFPXOWCKXUEKCA
|
9.7 | IC50 | 16 | — | |
KVKWRJDNIJTMGN
|
9.6 | IC50 | 16 | — | |
ZRKDDZBVSZLOFS
|
9.6 | Ki | 6 | — | |
WMBPDZBHEAETLZ
|
9.5 | Ki | 3 | — | |
RXMRVZANJZUNED
|
9.4 | Ki | 3 | — | |
RKXGEVUMNLOCDX
|
9.4 | Ki | 3 | — | |
QUUNMICPMYIHFS
|
9.4 | IC50 | 16 | — | |
VMDUABMKBUKKPG
|
9.4 | IC50 | 16 | — | |
WDCRWMNKRWOGOP
|
9.3 | Ki | 4 | — | |
RWUOGVWORJUNJA
|
9.3 | Ki | 4 | — | |
XKENJWNGLCKOBP
|
9.3 | IC50 | 16 | — | |
NJUMMJUUDUYSKB
|
9.3 | IC50 | 16 | — | |
ALBKMJDFBZVHAK
|
9.3 | IC50 | 16 | — | |
BYMDBFGHCDTBMT
|
9.3 | IC50 | 16 | — | |
IUHKSTINHDUYRO
|
9.3 | IC50 | 16 | — | |
VJVAWKPXJCDEQG
|
9.3 | IC50 | 16 | — | |
WRXDVVALWQGPMW
|
9.3 | IC50 | 16 | — | |
AJTIJRUGVRMRDN
|
9.3 | Ki | 5 | — | |
DHWTVCHLMXAWGK
|
9.3 | Ki | 3 | — | |
ULMLVGYYGWVNSC
|
9.3 | Ki | 3 | — | |
BUTCFAZTKZDYCN
|
9.3 | Ki | 6 | — | |
BLJPKQXXDFIIFR
|
9.2 | IC50 | 16 | — | |
XJMIBNLJFYSGAR
|
9.2 | IC50 | 16 | — | |
DLGWSCNXWHDMHZ
|
9.2 | Ki | 4 | — | |
KCEIOBKDDQAYCM
|
9.2 | Ki | 5 | — | |
JFGUJXZLJIUVPZ
|
9.1 | IC50 | 16 | — | |
LYFROTHEKIFZAU
|
9.1 | IC50 | 16 | — | |
RYIVVNHBYBYXHF
|
9.1 | IC50 | 16 | — | |
VZKRZUPJCVFVGR
|
9.1 | IC50 | 16 | — | |
DGBIGWXXNGSACT
|
9.1 | Ki | 16 | — | |
LHGSGTVATLBNGO
|
9.1 | Ki | 3 | — | |
YJZGQBGGTBIAOP
|
9.1 | IC50 | 16 | — | |
JYKXGGXAKPOFML
|
9.0 | Ki | 3 | — | |
AQKFCEWRKDXGMK
|
9.0 | Ki | 16 | — | |
FVFFDKKTXYVCCW
|
9.0 | IC50 | 16 | — | |
IPHSQMSRIWZULE
|
9.0 | Ki | 16 | — | |
KDMMIKQMHNBKAV
|
9.0 | Ki | 17 | — | |
KOVRZNUMIKACTB
|
9.0 | IC50 | 17 | — | |
RLFKILXOLJVUNF
|
9.0 | IC50 | 16 | — | |
WGRVAGIQTHEEQW
|
9.0 | IC50 | 16 | — | |
VREFGVBLTWBCJP
|
9.0 | Ki | 7 | — | |
BSBLYLUAUVTSMM
|
9.0 | IC50 | 16 | — | |
WQYYZNGOTUCWQX
|
8.9 | Ki | 5 | — | |
BQSIRVPTCKHWKR
|
8.8 | Ki | 5 | — |