Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
HRJQUDZTLASEPW 7.6 Ki 6
JXCPQLHXZUWOCZ 7.6 Ki 4
YMFJMRVJWVJJAB 7.6 Ki 5
HSUCRXNJMPDNOG 7.6 IC50 16
JNWDOTPNEZYWGO 7.6 Ki 16
NLHGXPUKOAOTRO 7.6 Ki 4
QNYDVDZHJMBNDK 7.6 Ki 2
QWWZARYPNGYPLG 7.6 Ki 3
XXVQXGKSBMSCHX 7.6 Ki 6
YTUMMZANIYQNOM 7.6 Ki 8
ZZTJJGWSKYVZIG 7.6 Ki 6
HCJVWLPVQMYLOI 7.6 Ki 8
JAFQEKAQGSQGTM 7.6 Ki 16
JYQBFIUGGKNLDH 7.6 Ki 6
KQTMWRZAVOUNCI 7.6 IC50 16
NFMFVESVKLVYJR 7.6 Ki 7
VIEKPLVJCPXIIB 7.6 IC50 16
XLKKKDPUVUIHEL 7.6 IC50 16
YKYOQIXTECBVBB 7.6 Ki 7
BTCSSZJGUNDROE 7.5 Ki 23
DLHLOWZPQSHARU 7.5 Ki 6
ICYHTUKXCNYVRM 7.5 Ki 6
RBWPBJRIJOEHCN 7.5 Ki 6
VXDPUKHUSNJVCJ 7.5 Ki 6
CDRADZRGYBTOKU 7.5 Ki 6
NUXNKKUXSDGYTN 7.5 Ki 7
WFCALMPXVKUYLO 7.5 Ki 3
AANJEGNNNSDLGW 7.5 Ki 16
AZIRFKLEFANUIC 7.5 Ki 6
PQAZYCAWLLSXHO 7.5 Ki 6
WDTGOYDHZIXMQO 7.5 Ki 7
WPJDKKSDGLIQQB 7.5 Ki 16
DRCGHGOPCPUYAI 7.5 IC50 16
IYEJMUDDGFBLEF 7.5 Ki 6
LTYUPBZLKIUGQX 7.5 Ki 8
NKIYALPHXLYICR 7.5 IC50 16
YOGKDBMNVNETRZ 7.5 Ki 6
FOSOKBNWILBLSN 7.5 Ki 16
INGJMHPGMVUEKY 7.5 Ki 6
KTFRBKXLNKKPEA 7.5 IC50 16
HRNSOLSYHZMSCD 7.5 Ki 6
ACVGNKYJVGNLIL 7.5 IC50 16
HYXFNGLXNMLTNQ 7.5 Ki 3
SCAPGUIFNHZJLH 7.5 IC50 16
SIPHVHFVEKBHKT 7.5 Ki 7
SUONVKFDJJYYME 7.5 IC50 16
AKDSPRXIQQMVKS 7.5 Ki 6
CRYMDEDOGKKRIT 7.5 Ki 6
MAZZBGKHYOJFSH 7.5 Ki 6
UKXDLKBYAPSHDL 7.5 Ki 6
2D structure