Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
BYEKIJACVDAPTD 7.7 Ki 16
LLAKESJIQFAQJA 7.7 IC50 16
OXUTXRZFYPFZEZ 7.7 Ki 6
QAMANTJYKWSLNP 7.7 Ki 6
ASUXILMTDDVWPD 7.7 Ki 7
FQDQLHDSVITISC 7.7 IC50 16
HKLYPSSDHPAOJM 7.7 IC50 16
HRVCUISAJOBFTQ 7.7 Ki 6
NDFKYGUTDGWIHX 7.7 Ki 6
RSEMKXACIMVTQP 7.7 Ki 16
QOICRVBHAUSMFA 7.7 Ki 6
WDTNKNNGHGOKBH 7.7 Ki 9
WRDHNUVAWMYMJK 7.7 IC50 16
AURFZBICLPNKBZ 7.7 IC50 16
GWZLKOYBOFFDEB 7.7 Ki 6
NLEQOPYBIKKOPK 7.7 Ki 7
PSDFROGPPFTBND 7.7 Ki 7
RBMPSWHARBABOC 7.7 Ki 6
ZFLBRINMIQTFNB 7.7 Ki 18
WLZXRXFLGSQYFP 7.7 Ki 4
BPKZCNBWMWKTIB 7.6 Ki 4
CJYPUCKDMBCYEH 7.6 IC50 16
GGSVEKWMDFBTDG 7.6 Ki 4
HBBBENORIXSUJV 7.6 Ki 6
LNPSYDJGQQETLB 7.6 Ki 16
TWQDMCPDTPVCQP 7.6 IC50 16
VHQCVUYEMJHQEX 7.6 Ki 16
XQXQETQWDXIRQS 7.6 Ki 2
UFSSPXFMMJZZDU 7.6 Ki 4
CBAXLHGEEASOPH 7.6 Ki 6
CVNPFPRAINQAHI 7.6 Ki 5
FUTRDVKMGNYUPP 7.6 Ki 6
IDTSXEWVFBEMPN 7.6 Ki 6
JHDNCJGODWCHES 7.6 IC50 16
LIXHLXZPUZQKCT 7.6 IC50 16
LLJUUCOIBTZXIJ 7.6 Ki 6
PDOZRVXKPBQAJH 7.6 IC50 16
RZXWKGHDRQNABH 7.6 IC50 4
VVBYXJYBLBPAEN 7.6 Ki 6
JWLCOGXPTWMMDY 7.6 Ki 16
UPPLJERIZONGME 7.6 Ki 6
CMUJABAHLCISIQ 7.6 Ki 6
FNNPSIGQQWCKKB 7.6 Ki 5
KBVJZOBCOIANOX 7.6 Ki 16
KOMBGWPXIHBMLL 7.6 IC50 16
MBBOXTKOOFAZLI 7.6 Ki 16
OSHQANHMWJQRHB 7.6 Ki 16
RTHSDLLYNWWMSZ 7.6 Ki 6
ULMKSNRBNFFOJQ 7.6 Ki 16
ZWJGDMSWCKASII 7.6 IC50 16
2D structure