Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
QGOAGGOYLMIFPI 8.0 Ki 6
HGJUDXDUSGEVOX 8.0 Ki 6
HQJSGBKPXYZTRN 8.0 IC50 16
JEUGTSHICBOMGA 8.0 Ki 3
MBZNSAJBODIJCK 8.0 IC50 16
OJVFFZLXISLIFZ 8.0 Ki 6
YVAHCWLEKOONFT 8.0 Ki 3
IAIZAMKHEDKXAK 8.0 Ki 6
RJOMRLSAWXNFSU 8.0 Ki 4
GAONFNHSQRTFJA 8.0 Ki 6
HFPZDEHIDKJZSN 8.0 Ki 16
IBPJOIOGTFGBRO 8.0 Ki 6
IXGIOXIKQZCZIK 8.0 Ki 8
JTYYMOMTGZSRFM 8.0 IC50 16
LMJMBPXKXWIKQK 8.0 IC50 16
NNHRCSJWUBQYQV 8.0 IC50 16
PKJGSRHYDOGGLB 8.0 Ki 17
PYXJKYJAFMLYMS 8.0 Ki 6
YVPJMZCJVHJOFG 8.0 Ki 7
FJLMOGVUSSSKEC 7.9 Ki 16
LLAKESJIQFAQJA 7.9 IC50 16
ZDGLRCMEFVYZHG 7.9 Ki 6
CNFLHWVYIFARIM 7.9 Ki 7
CNVQMRWAJHEFGZ 7.9 Ki 16
CUICGHSKDSXIRX 7.9 Ki 6
IEDCFFRFAIAYGF 7.9 Ki 7
MZTRNWROWIGTRB 7.9 Ki 7
OPMIQGMTRGXAQY 7.9 IC50 16
VAARLVBAANTQOM 7.9 Ki 16
YVTIEXKHDRKBSM 7.9 IC50 4
ZWWXXHQAJKCRDM 7.9 Ki 6
CLMNGHYEDSVQIK 7.9 Ki 6
GXYIMPYRUIKXIS 7.9 Ki 6
HSEWUGOOPIEKBZ 7.9 IC50 16
PBUYINIRVVLBIH 7.9 Ki 4
SUBCTDHFKBVAQE 7.9 Ki 3
UNJFTNACNPGPEC 7.9 Ki 6
XAMVDLCXXPEEEG 7.9 Ki 16
XUJMJGTVTZESCM 7.9 Ki 7
RJNFLJNUEOERRU 7.9 Ki 6
YLRURIRIQRAQJJ 7.9 Ki 16
MVCCGUFWBDSIHW 7.9 Ki 3
DXSIUJMZGGYSFI 7.9 Ki 3
NHJFEXZXSCFYRX 7.9 Ki 6
RFNXMSGJCRYTIU 7.9 Ki 3
XGEQEYJHZCAALH 7.9 Ki 3
PZIQTZQOFYKORR 7.8 Ki 6
WAEXHEOACCAOSS 7.8 Ki 16
YLPHFEFMBAMSKS 7.8 Ki 5
GADIKQPUNWAMEB 7.8 Ki 5
2D structure