Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
GTGGDPMSPFTXEJ 8.2 Ki 3
BDISWVKOOATATE 8.2 Ki 16
PCRRXYJDKILUID 8.2 Ki 6
HLKQVESZETYPOB 8.2 Ki 3
YJQPSUGEFJEJIN 8.2 Ki 6
YUOOYQDBXTWPKL 8.2 Ki 16
ACUNYYFYYWOKOD 8.2 IC50 16
CDWXZILKRXSANI 8.2 IC50 16
MSYBIYCNXBCGOA 8.2 Ki 2
QIZPCEVRKTWHIE 8.2 IC50 16
OTQXKRRISJPTFS 8.2 IC50 16
SNVZCVVNVLIROS 8.2 Ki 6
WMCJJXHYPNOCMT 8.2 IC50 16
ZRPUPUBWCXFOCY 8.2 Ki 16
LCNUELABLMGVTP 8.1 Ki 3
LJRIFLWERUHAIZ 8.1 Ki 8
MMBJQNHQQHDAKU 8.1 Ki 3
NESUAJPAOMXMJC 8.1 Ki 6
JOHKRJNYKDHTID 8.1 Ki 6
SSJXJXJUHUAOQL 8.1 Ki 6
VQAWSSJLGHVFHE 8.1 Ki 6
DKCAUMRZSZVJCP 8.1 Ki 16
IVGTVZGLPHBTJV 8.1 IC50 16
IVGTVZGLPHBTJV 8.1 IC50 16
JSDYTEOPJOVCPM 8.1 Ki 6
NHJRHDMRNNOSLV 8.1 Ki 5
OSMYMXKHKOTLKC 8.1 Ki 7
QVIQGNJPFOVZBZ 8.1 Ki 16
YHNNMZUUFMJQQY 8.1 IC50 16
DXPCEAZKJSYFJM 8.1 Ki 6
YNPDBSCCAHYJAP 8.1 Ki 2
TWSTVDPXWQPIIM 8.1 Ki 4
ZCQOZHJHIVMMEC 8.1 Ki 2
MMWKMKRWCPKFRA 8.1 Ki 6
VBXZLYYHFDVNEN 8.1 Ki 6
VOVGYBOEGUOGJQ 8.1 Ki 3
XNIDSAVZEZPOBT 8.1 Ki 6
FLTOAJWVMNMXMX 8.1 Ki 6
NVWCZRPXYVDQEE 8.1 Ki 5
ACHPNNOYBNCORU 8.1 Ki 8
ACVGNKYJVGNLIL 8.1 Ki 5
IACRYXFWKJOMEI 8.1 Ki 3
XGJLRKVQXMSBJW 8.1 IC50 16
HJNOESUOZGNLKO 8.0 Ki 6
ZJQHPWUVQPJPQT 8.0 Ki 17
FLEQTIDRWGGTRR 8.0 Ki 7
DQGKGLFOXZGWHX 8.0 Ki 2
HEGJYRQUDMITRQ 8.0 Ki 6
KWPOKTUWXDCATM 8.0 IC50 16
OBPPXGLDCMXNDT 8.0 Ki 6
2D structure