Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
IVVHFTRDYKTGCC 8.4 Ki 6
MVBVNOZDVRVMNH 8.4 IC50 16
GFQMHVYMEKXHDT 8.4 Ki 6
OKGJPMZATLJSGV 8.4 Ki 6
WLHRDALLBOSVLX 8.4 Ki 6
AXPGZURVLRWNBR 8.4 Ki 16
BZVWONIGXAYZIT 8.4 IC50 16
DYSDYZCGZCYPCT 8.4 IC50 16
LMXUGQJMQSMLIQ 8.4 Ki 17
MFZNONRIQYSLMZ 8.4 Ki 6
UULFOYXSWNADTF 8.4 IC50 16
ALBKMJDFBZVHAK 8.4 Ki 16
MKNXZRAKHYWDOS 8.4 IC50 16
VCPRTCGXKBSFJJ 8.4 Ki 4
XQUJTESAXUTXNH 8.4 Ki 16
BWWQXKSOWUMHAQ 8.4 Ki 6
RLFKILXOLJVUNF 8.4 Ki 16
CFMPKKXOXYNZHF 8.3 Ki 6
AHHSTGLUTRNWRJ 8.3 Ki 6
KBMIXEOSQPPORV 8.3 Ki 8
IPRPEMNPDVAAOU 8.3 Ki 3
YGKSPOBIXHTPMV 8.3 IC50 16
KOVRZNUMIKACTB 8.3 Ki 17
QWWODAPIEHJFQG 8.3 Ki 16
ACMQMUZDLQDWTK 8.3 Ki 16
GOCZPCXRIJMRNR 8.3 Ki 16
HTNYBQDFFUZWCY 8.3 Ki 5
PHOATQSOBKATTD 8.3 Ki 16
PTRXPVDOTUGGHW 8.3 IC50 16
UKHFPVCOXBJPIN 8.3 Ki 17
DKSWXNFPYZCJFU 8.3 Ki 6
MZGKIGRVCYKVPS 8.3 Ki 6
AOZALWRGTMILIK 8.3 Ki 6
XBPAHSBPWSBJHT 8.3 Ki 6
NTSIBLRVVRGOLO 8.3 Ki 3
ZWWZTFYQCITUTK 8.3 IC50 16
GIISEXDJPQATBL 8.2 Ki 2
SJAGJFDQMIAULO 8.2 Ki 6
BGGCZORPGAXQJX 8.2 Ki 3
DZPQKPSHACGLKC 8.2 Ki 6
ZDLKXIOQJJRYCW 8.2 Ki 6
KSYVJHGNJMYDIQ 8.2 Ki 6
BTLWEEGNXUJKKB 8.2 IC50 16
KIVQXKXZISOGBE 8.2 Ki 17
NKIYALPHXLYICR 8.2 IC50 16
OKKCDBHXMZEFNG 8.2 Ki 3
VIILRVHOGYZXSZ 8.2 Ki 2
YUSWMAULDXZHPY 8.2 Ki 20
ZRRVSALMQDOQAX 8.2 Ki 16
BGRWSFIQQPVEML 8.2 Ki 6
2D structure