Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
JMRHVJPVNLBGRZ 8.7 Ki 3
RLLAIMNJXRQPNZ 8.7 Ki 2
AAFXZNIGLSLXPH 8.7 IC50 2
HNGRWUCKESPKRC 8.7 Ki 6
LRHBSPDBIHZAOV 8.7 Ki 2
OTWGFFXBGMUFBP 8.7 Ki 6
YKKWBLSUYZOORV 8.7 Ki 6
GTOBFJHFOZIFFU 8.7 Ki 5
SEWXZWMBVGJJPG 8.7 Ki 7
VMDKDKVHHDTDAL 8.7 Ki 4
KXZNTMNIMNTHIP 8.7 Ki 2
OVXGOBUGGHQLKJ 8.7 Ki 2
QTEUJQNPMLXVLL 8.7 IC50 16
VJMXGRAYTDRKAO 8.7 Ki 6
VHGIDFXNMYWNMX 8.7 Ki 3
CHMFFBQMSYJXTP 8.6 Ki 6
LDRJMZJUSNJPQM 8.6 Ki 2
QSEBFHRZNPGODU 8.6 Ki 6
RZOFEWOHNOOHND 8.6 Ki 6
ZOCSXAVNDGMNBV 8.6 IC50 16
NRBRKRZMKXLHTR 8.6 Ki 3
PPTYJKAXVCCBDU 8.6 Ki 7
ZQLPLWRQUVVKJZ 8.6 Ki 6
LHMYCKKRCBXCBI 8.6 Ki 5
CWDNSPMTRZUBER 8.6 Ki 2
CHIFCDOIPRCHCF 8.6 IC50 16
CHQPOBHNDRMXFK 8.6 Ki 18
LSVOXYMZIGSSNB 8.6 Ki 6
VAJLZGPUVKNCRO 8.6 Ki 6
VXVLSQVFRWSMKF 8.6 Ki 6
ZKVGHURGXXUFQB 8.6 Ki 6
AHTXTFPELOVMKB 8.5 Ki 6
HOQUSTXYXSUJDG 8.5 Ki 6
OIVNHVRINWMDTH 8.5 Ki 5
QPBUEBDNKGGQCP 8.5 Ki 3
STHRYAZDXIDVJO 8.5 Ki 6
KVKYGVOAHGNAKZ 8.5 IC50 17
LENHHZQGSWCZJW 8.5 Ki 16
NEOUOHDNZDRDNJ 8.5 IC50 16
RYLDZJANGRBUGW 8.5 IC50 16
YMEKUDZYTKIXGP 8.5 Ki 2
DKGPQXLYULZUKP 8.5 Ki 2
JRCQRBJGHBZPRG 8.5 Ki 3
AWOOMIRCBITDFK 8.5 Ki 6
SSTBAKDUFHYWMX 8.5 Ki 2
YWVNAIWRDXBOOS 8.5 Ki 6
PFJHXYJLEIZLGQ 8.5 Ki 6
QBYZDDIMNITMSB 8.5 Ki 6
KADHNYOMTSABQA 8.4 Ki 3
DTUMUPWQPZERNQ 8.4 Ki 2
2D structure