Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
OFBIFZUFASYYRE 9.1 Ki 16
YJZGQBGGTBIAOP 9.1 IC50 16
BPTASZCHRIMWEF 9.0 Ki 6
UIBMSUDAMPUYHS 9.0 Ki 2
AQKFCEWRKDXGMK 9.0 Ki 16
BQSIRVPTCKHWKR 9.0 Ki 5
BUTCFAZTKZDYCN 9.0 Ki 6
DVVOGWYOYHNNQP 9.0 Ki 3
IPHSQMSRIWZULE 9.0 Ki 16
KDMMIKQMHNBKAV 9.0 Ki 17
OGBTVLIUFUJHTH 9.0 Ki 5
OXDLZFDSMXMUKS 9.0 Ki 3
QXZGSQAJHBQSSV 9.0 Ki 4
WGRVAGIQTHEEQW 9.0 IC50 16
BSBLYLUAUVTSMM 9.0 IC50 16
WEFRNUXPTYTOEU 8.9 Ki 3
ASOMQCZKXCZAAQ 8.9 Ki 2
BNQJKHFCSDKTCD 8.9 Ki 4
DGBIGWXXNGSACT 8.9 Ki 16
IRYAGFJMRZLHGE 8.9 Ki 6
KKWDMTXJUXKNOU 8.9 Ki 7
LWUDDYHYYNNIQI 8.9 Ki 6
PELQRWYXKWRIDE 8.9 Ki 2
UFTKNTUWDMJOIX 8.9 Ki 16
WRXDVVALWQGPMW 8.9 Ki 16
IUHKSTINHDUYRO 8.9 IC50 16
MKQJGNJLLCPKEB 8.9 Ki 2
KOOUQKARBNOFGH 8.8 Ki 2
PEEGZDFBOLCRFF 8.8 Ki 4
YTGZSWOWFGVAFH 8.8 Ki 7
XJMIBNLJFYSGAR 8.8 IC50 16
YLDRVNNGBACDSD 8.8 Ki 6
BJYKRVMKNGJKKZ 8.8 Ki 6
OLKUNPKISSHQBO 8.8 Ki 6
VJVAWKPXJCDEQG 8.8 IC50 16
PFZUQESQYBPRGB 8.8 Ki 3
UWQBBGFHDXOYNN 8.8 Ki 2
XTZAPIKNFFKUDJ 8.8 Ki 2
FTBGMXWQYKNAKT 8.8 Ki 6
FYOXWZFDOADHOW 8.8 Ki 6
HEFBZEKZYFOEGG 8.8 Ki 2
OJLYUGSSUKAWJC 8.8 Ki 16
QZDWWRKBDPYMIP 8.8 Ki 6
RGDHMJMNRYQXCW 8.8 Ki 6
KVKYGVOAHGNAKZ 8.7 IC50 16
NURMFSYNABAOFU 8.7 Ki 6
VKXOQBAHWPYQGS 8.7 Ki 2
CLKDKLQSBMZIQH 8.7 Ki 2
PCZLQMGFNUNVOM 8.7 Ki 6
ZPSBXQBYCQOCEU 8.7 Ki 6
2D structure