Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
NRCNHRJESVKFJO 7.2 Ki 6
SNBBNIBMHQGUBE 7.2 Ki 7
BTESADIOSMFPBT 7.2 Ki 6
NKSQLOHZBFUKLF 7.2 IC50 16
RCPDOEFGDWHVCA 7.2 Ki 6
CAIDJZOHDFNJOZ 7.2 Ki 4
LIIRYFLHPZDMEC 7.2 Ki 6
OEIRQQZGARGKRG 7.2 Ki 6
PRUQRKPURHYKRP 7.2 Ki 16
VAVBWHIBLOPOEM 7.2 Ki 16
BULOMLIWEVCBPE 7.2 Ki 6
IOOGUHXPDYRXFJ 7.2 IC50 16
ANKFABXSPKCYOQ 7.2 Ki 6
GZPJZUILYCOUHJ 7.2 Ki 6
WCYJVRQPVHPWLQ 7.2 Ki 16
WHEUGJHMVJCNEP 7.2 IC50 16
KICQPTHJQWBQOI 7.2 Ki 7
SINAJPKUKOSXOT 7.2 IC50 16
YHHCQFOSZRZNQC 7.2 Ki 5
KPKJEFIYLPVANT 7.2 Ki 4
LPOZDKMXSPAATL 7.2 Ki 16
PRGDQIDWABTGRF 7.2 Ki 4
MDTMAWZEUAVCQZ 7.1 Ki 6
XHXRMYICRMVHBK 7.1 Ki 4
ZRZOZCBSSVQEGD 7.1 Ki 6
KUZLDKPQBCXMLJ 7.1 Ki 6
VOZOMZWSLGQRKP 7.1 IC50 16
SZDYQTCZTLGXBX 7.1 Ki 6
YBRXFNLNMSTVNQ 7.1 IC50 16
YKVBFMDDXCMYHI 7.1 Ki 5
DXCKAYBKZBTPNN 7.1 Ki 6
IKXSFQFVTQDDAR 7.1 Ki 6
HOXKKBLQXUBSEI 7.1 Ki 6
HRTSOMLTEJFUCO 7.1 IC50 16
PGTVWKLGGCQMBR 7.1 IC50 16
KBFYDAGNYWSKLZ 7.1 Ki 6
LQKOTGTWBANJBS 7.1 Ki 6
OMQHFPMEAPEGTA 7.1 Ki 16
VJXWQJKLMZXRCW 7.1 Ki 6
GSJSXDQXHDAYLZ 7.1 Ki 6
KJUPZRXGDNYFQT 7.1 Ki 6
YSURNJBIVZXADU 7.1 Ki 5
ZSMNMYCBVFAPQG 7.1 Ki 6
BOVVCNDNINYMTL 7.1 Ki 6
KDGMRQJYYKGVCJ 7.1 Ki 7
AEYRTFCCYIWUJJ 7.1 Ki 16
LOFKMRMDVCEZEF 7.1 Ki 7
NFXAWQDTYKJJTD 7.1 IC50 16
JSRKYARWMIOKOB 7.0 Ki 16
LWLYOXPDYPYNHH 7.0 IC50 16
2D structure