Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
SZHAAZHKMCGJJK 7.3 Ki 4
GWCQPEHFUKZODL 7.3 Ki 16
CAJUSRIHDIZNNF 7.3 Ki 6
DRCWBQAOFNLXIV 7.3 Ki 7
HRUDFUBJGCKXQF 7.3 Ki 6
BALGGUJCACDSLM 7.3 Ki 6
NCOMRCAHJHWHOU 7.3 Ki 4
QYEIQYJLVREYBI 7.3 IC50 16
RELKUIIVWKRWEL 7.3 Ki 7
SIBRGSBVGDWJAF 7.3 IC50 16
WHGIBMIKSVYLCR 7.3 IC50 16
ZYQKNGNVEVNORP 7.3 Ki 6
AURFZBICLPNKBZ 7.3 IC50 16
COKSTUDOWROCJE 7.3 Ki 6
DGZYPGWWTKGBQP 7.3 Ki 16
DVKHCFDZNVGRQT 7.3 Ki 16
LPAODQAWVMEXKR 7.3 Ki 16
NTZNKZHCQIJCPO 7.3 IC50 16
QAXDJUNLAJMPAE 7.3 Ki 6
SNEWVMXJSABDSK 7.3 Ki 16
VWCCHJFFYCGXFL 7.3 Ki 16
JBDRNSFDKSBSFE 7.3 Ki 16
NNHRCSJWUBQYQV 7.3 IC50 16
OGZWYHFVQMYPED 7.3 Ki 6
PISRVNOAPOPQHJ 7.3 Ki 18
DLEWDNHPWLPKDJ 7.3 Ki 8
GQIVRYNNTCEOBX 7.3 Ki 8
KRVDMABBKYMBHG 7.3 Ki 16
VOZOMZWSLGQRKP 7.3 IC50 16
XEJHLKHWRSNEOC 7.3 IC50 16
DSTVUBPAEXKNMB 7.2 Ki 6
KPKJEFIYLPVANT 7.2 Ki 4
MVMSIAOIXGSGIK 7.2 Ki 3
QBWJMTOHSYOPBE 7.2 Ki 7
UEWSJGMYAPQKKT 7.2 Ki 16
ULDBOWIRGDMZPF 7.2 Ki 8
URMNROOZTOLUHQ 7.2 Ki 16
YMIKAQYPFQWUEM 7.2 Ki 7
YTPPBAYYHIGVLQ 7.2 Ki 3
MGVMCBAQXDZWTN 7.2 Ki 6
PWOQCZLPANHRRJ 7.2 Ki 16
SFQDQVWLPSONMD 7.2 Ki 6
YNGRKYAIISTAOT 7.2 IC50 2
ZAFFVUHUTAMYCX 7.2 Ki 6
AYRJXCIMSHQLPG 7.2 Ki 6
HRNSOLSYHZMSCD 7.2 Ki 5
KZSDRHSSHPIBAO 7.2 Ki 6
GJGYQBVUXZXJSO 7.2 Ki 5
HRNSOLSYHZMSCD 7.2 Ki 6
LFWNCDNFYFPIPT 7.2 Ki 3
2D structure