Target not found.
Target not found.
Target Details
UniProt ACP47869
Gene SymbolGABRA2
Protein NameGamma-aminobutyric acid receptor subunit alpha-2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 901
  • Clinical molecules 0
  • Avg pChEMBL 7.52
Top Co-occurrence Targets
Active Molecules (901)
InChIKey pChEMBL Type Targets Clinical
CGMJQQJSWIRRRL 10.2 Ki 6
ZRKDDZBVSZLOFS 9.8 Ki 6
MZFKWSFOAVBLQM 9.8 IC50 16
QUUNMICPMYIHFS 9.8 IC50 16
WFPXOWCKXUEKCA 9.7 IC50 16
VTXIBIOXWRGGBL 9.6 Ki 2
KVKWRJDNIJTMGN 9.6 IC50 16
VACJUKKURQMWHE 9.6 Ki 5
NTQIDFIQUNKLIH 9.5 Ki 5
QKIWQBLNTSQOLY 9.5 Ki 6
QVMKXYFWXJHPIX 9.5 Ki 2
UZZBNSRTLAFTLY 9.5 Ki 2
KYDURMHFWXCKMW 9.5 Ki 6
FGOCJZANGVRDDB 9.4 Ki 3
UAISVGZOWWUBIG 9.4 Ki 2
UMBHXQNJEMMKIG 9.4 Ki 3
JGVFVEUZTKIPIB 9.3 Ki 2
XKENJWNGLCKOBP 9.3 IC50 16
BJDIHPUUUSHMRK 9.3 Ki 2
NJUMMJUUDUYSKB 9.3 IC50 16
NVETZYIXXYETLA 9.3 Ki 6
DSDYDTCIWBGXBT 9.2 Ki 2
KJDDJAPSHCVDDC 9.2 Ki 3
PEBWTLIJBCZFOA 9.2 Ki 6
NZMJFRXKGUCYNP 9.2 Ki 6
JOFWLTCLBGQGBO 9.2 Ki 8
OWOWBGNEZCVQKU 9.2 Ki 2
VXSLAFXNESWHFV 9.2 Ki 2
BLJPKQXXDFIIFR 9.2 IC50 16
LOZNAQDBHKVLRN 9.2 Ki 6
SRAWBNFSMIHBEM 9.2 Ki 8
VREFGVBLTWBCJP 9.2 Ki 7
JNJUWXAKLRKXII 9.2 Ki 6
LWUDDYHYYNNIQI 9.2 Ki 7
NPISRJOTBMWCDJ 9.2 Ki 2
QGMKNRLNMKUUEC 9.2 Ki 2
BQDUNOMMYOKHEP 9.2 Ki 6
BYMDBFGHCDTBMT 9.2 IC50 16
KCEIOBKDDQAYCM 9.2 Ki 5
UWXAQZGCSSYTJL 9.2 Ki 6
CMSKDYKEKYIJSD 9.1 Ki 5
ISZRIZPRXUQOMU 9.1 Ki 5
BCLNCXBDWXPRAH 9.1 Ki 4
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
VZKRZUPJCVFVGR 9.1 IC50 16
QYSYOGCIDRANAR 9.1 Ki 7
XXRKXVKJMSIZSM 9.1 Ki 6
GMMRKZMQEHKQPX 9.1 Ki 2
2D structure