Target Details
| UniProt AC | P46937 |
|---|---|
| Gene Symbol | YAP1 |
| Protein Name | Transcriptional coactivator YAP1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF15238 (TEADIR3) PF00397 (WW) |
Summary
- Multi-target molecules 18
- Clinical molecules 0
- Avg pChEMBL 6.87
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLCVDQHLYHBAHR
|
9.0 | IC50 | 2 | — | |
QRAZSFFSGBFSLJ
|
7.7 | IC50 | 2 | — | |
FMFQQQHCFDLITQ
|
7.6 | IC50 | 2 | — | |
VVQSZBAMNWEOFA
|
7.4 | IC50 | 2 | — | |
KRSSVRNWESYFMZ
|
7.1 | IC50 | 2 | — | |
RHLHNRVWVMXZTL
|
7.1 | IC50 | 2 | — | |
DJGXOJSWOLDZPW
|
7.1 | IC50 | 4 | — | |
MRLLZKOSLONRSI
|
7.1 | IC50 | 5 | — | |
JLFVYIWUQHPMTB
|
6.7 | Kd | 2 | — | |
RRBNTBZUGZSZPY
|
6.5 | IC50 | 2 | — | |
LBTWZXYXMWBYRV
|
6.5 | IC50 | 2 | — | |
JJKYNQHCVCQSIQ
|
6.5 | IC50 | 2 | — | |
GAQQHLRNBQSZHG
|
6.4 | IC50 | 2 | — | |
FRCDQCXLBBSGID
|
6.4 | IC50 | 2 | — | |
VMZAMOYHCUWUAW
|
6.3 | IC50 | 2 | — | |
CVZOMJMMROGASZ
|
6.2 | IC50 | 2 | — | |
GGXKLNSXPSGXJU
|
6.0 | IC50 | 2 | — | |
JGIYBKFOIUVCQB
|
6.0 | IC50 | 2 | — |