Target Details
| UniProt AC | P46925 |
|---|---|
| Gene Symbol | PMII |
| Protein Name | Plasmepsin II |
| Organism | Plasmodium falciparum (isolate HB3) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00026 (Asp) |
Summary
- Multi-target molecules 220
- Clinical molecules 0
- Avg pChEMBL 7.17
Active Molecules (220)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YFZWFIKCKDMMME
|
6.2 | Ki | 2 | — | |
AWCGJEFUHUSFBQ
|
6.2 | IC50 | 2 | — | |
LAHQEHNTHAUTTK
|
6.2 | Ki | 2 | — | |
LOBCJUCVSNWELD
|
6.2 | IC50 | 3 | — | |
TUYZMTOTGANLMU
|
6.2 | Ki | 2 | — | |
NCNMSGOJBLVCOM
|
6.1 | IC50 | 3 | — | |
CSWMOEBFXLXGOK
|
6.1 | IC50 | 2 | — | |
DOFWARZRCWUXKJ
|
6.1 | Ki | 2 | — | |
VEWFKNUERSAOIS
|
6.1 | IC50 | 3 | — | |
PZCSYTKHAKPNOQ
|
6.1 | Ki | 2 | — | |
NKSLZHUZXVIXOR
|
6.1 | IC50 | 4 | — | |
WDKZPITZRFMOHK
|
6.0 | IC50 | 3 | — | |
FCCCRBDJBTVFSJ
|
6.0 | IC50 | 2 | — | |
LYGGDXLOJMNFBV
|
6.0 | IC50 | 2 | — | |
NJBBLOIWMSYVCQ
|
6.0 | Ki | 3 | — | |
OFMNXXZKHSYCMQ
|
6.0 | IC50 | 2 | — | |
PNSQCPQDRVOKMA
|
6.0 | IC50 | 2 | — | |
QMGXWNSSMGAHCA
|
6.0 | IC50 | 2 | — | |
YBBSKAGTEPBSNK
|
6.0 | IC50 | 2 | — | |
YBQZXXMEJHZYMB
|
6.0 | IC50 | 2 | — |