Target Details
| UniProt AC | P46663 |
|---|---|
| Gene Symbol | BDKRB1 |
| Protein Name | B1 bradykinin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 88
- Clinical molecules 24
- Avg pChEMBL 8.26
KEGG Pathways (6)
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WPZQFRGWZRSMKV
|
8.0 | IC50 | 2 | — | |
UFPMXLUTBQTILN
|
8.0 | IC50 | 2 | — | |
RQIRBNSHBCLESE
|
8.0 | IC50 | 2 | — | |
IQUDIMJYXGNLDC
|
8.0 | IC50 | 2 | — | |
SDJNJNHVRLVGFW
|
7.9 | IC50 | 2 | — | |
IAWVOODBIZSXKE
|
7.9 | IC50 | 2 | — | |
MFMVOZVJMLNPKU
|
7.9 | IC50 | 2 | — | |
DHXMASVOPVPEJZ
|
7.8 | pIC50 | 2 | Yes | |
IIMPAUOPPFMYKX
|
7.7 | IC50 | 2 | — | |
YOFLVURHBHANJB
|
7.6 | IC50 | 2 | — | |
FDNSGRXVGYVALV
|
7.5 | pIC50 | 2 | Yes | |
KLNCTQVQTQNZGS
|
7.5 | IC50 | 2 | — | |
UQNOVFWEEACSGU
|
7.5 | pIC50 | 2 | Yes | |
BLGPUKWHJXZTPQ
|
7.4 | IC50 | 2 | — | |
FDNSGRXVGYVALV
|
7.4 | pIC50 | 2 | Yes | |
MDVKPFWDLCCUPM
|
7.2 | pIC50 | 2 | Yes | |
RBIXVHPHNGXTCI
|
7.2 | pIC50 | 2 | Yes | |
ULEVRJKNZJLMMK
|
7.2 | IC50 | 2 | — | |
YCYBPINOGLKAOI
|
7.2 | IC50 | 2 | — | |
BRUUOQFUWNUOGV
|
7.1 | IC50 | 2 | — | |
MBIKZIVONJGCJQ
|
7.1 | IC50 | 2 | — | |
YMROZBYZFLPAPA
|
7.1 | Ki | 2 | — | |
WRPSCMJWFRBZKH
|
7.0 | pIC50 | 2 | Yes | |
CHXHGDPPQTWZQN
|
7.0 | IC50 | 2 | — | |
MDKZHOJYEIZDMH
|
6.9 | IC50 | 2 | — | |
VWEXBIUSTBETLM
|
6.9 | IC50 | 2 | — | |
KULRZBJHHZWTME
|
6.8 | pIC50 | 2 | Yes | |
OZETVGJPQDGYFE
|
6.7 | IC50 | 2 | — | |
DHSJWRXSMQPZKV
|
6.6 | IC50 | 2 | — | |
RIOBXZSQDXGNJE
|
6.6 | IC50 | 2 | — | |
IQEQRSGEGRUUMU
|
6.4 | IC50 | 2 | — | |
MTFMCHRVVYXNMF
|
6.4 | IC50 | 2 | — | |
STNBXDIHDUXATH
|
6.4 | IC50 | 2 | — | |
XQRBXNACKNDXEL
|
6.3 | IC50 | 2 | — | |
NELJVFSIQMBCNA
|
6.2 | IC50 | 2 | — | |
WBBTXKGNCKTYFN
|
6.2 | pIC50 | 2 | Yes | |
CJKSFDBEHUXSSN
|
Clinical | TTD_MultiTarget | 2 | Yes | |
DRZRLKNZUGAIDL
|
Clinical | TTD_MultiTarget | 2 | Yes |