Target Details
| UniProt AC | P46663 |
|---|---|
| Gene Symbol | BDKRB1 |
| Protein Name | B1 bradykinin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 88
- Clinical molecules 24
- Avg pChEMBL 8.26
KEGG Pathways (6)
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QXZGBUJJYSLZLT
|
11.0 | pIC50 | 2 | Yes | |
DSKXSKYPLRUWNI
|
10.6 | Ki | 2 | Yes | |
DSKXSKYPLRUWNI
|
10.6 | Ki | 2 | — | |
DSKXSKYPLRUWNI
|
10.6 | Ki | 2 | Yes | |
PWPVANGLZUNDSV
|
10.5 | Ki | 2 | Yes | |
PWPVANGLZUNDSV
|
10.5 | Ki | 2 | — | |
SKEDKPUBPAWRPO
|
9.8 | pIC50 | 2 | Yes | |
UXMVCNAZMAVIBE
|
9.7 | Ki | 2 | Yes | |
PAUIXIOLYSEIEG
|
9.2 | IC50 | 2 | — | |
KYOLIWRJBMRTOA
|
9.2 | IC50 | 2 | — | |
WJLDXLVGJQBDFE
|
9.1 | IC50 | 2 | — | |
KULRZBJHHZWTME
|
9.1 | pIC50 | 2 | Yes | |
QDFIXHJNZHRIQL
|
9.1 | IC50 | 2 | — | |
SNCVXRFWMPIJGT
|
9.1 | IC50 | 2 | — | |
HOONOQPHTXFQCK
|
9.0 | IC50 | 2 | — | |
MNSIVJGXSIVXGB
|
9.0 | IC50 | 2 | — | |
QIUGDRUGWFFHGP
|
9.0 | IC50 | 2 | — | |
MDVKPFWDLCCUPM
|
9.0 | pIC50 | 2 | Yes | |
WBBTXKGNCKTYFN
|
9.0 | pIC50 | 2 | Yes | |
WBBTXKGNCKTYFN
|
9.0 | pIC50 | 2 | Yes | |
MIJKUFVQFDMZAW
|
9.0 | IC50 | 2 | — | |
WGIMYCFLPCKLAB
|
9.0 | IC50 | 2 | — | |
RDGDPEKYNKOHFV
|
9.0 | IC50 | 2 | — | |
FNFMOUAVCVSXID
|
8.9 | IC50 | 2 | — | |
RYMCKAQYHQAPMB
|
8.9 | IC50 | 2 | — | |
FNLYZFQVRYPOPT
|
8.9 | IC50 | 2 | — | |
OFBIENNCBQWFEJ
|
8.9 | IC50 | 2 | — | |
HMJOZKNMJKJYHS
|
8.8 | IC50 | 2 | — | |
KFDYGIUPQPPPND
|
8.8 | Ki | 2 | — | |
QNVIMPQAFIYICG
|
8.8 | IC50 | 2 | — | |
DNZZUJBLUHTHMB
|
8.8 | IC50 | 2 | — | |
IJUBQVLOLZAVCN
|
8.7 | IC50 | 2 | — | |
HJCJUXBDBHUVCI
|
8.7 | IC50 | 2 | — | |
LXQWSJLJIHTFOW
|
8.7 | IC50 | 2 | — | |
CIQDQPSLIUICPX
|
8.7 | IC50 | 2 | — | |
WRPSCMJWFRBZKH
|
8.7 | pIC50 | 2 | Yes | |
JKQWZANTQIVDTL
|
8.7 | IC50 | 2 | — | |
JRXMTRHRQJCCHA
|
8.6 | IC50 | 2 | — | |
RLZPVLDPNQNXFY
|
8.6 | IC50 | 2 | — | |
CJKSFDBEHUXSSN
|
8.6 | pIC50 | 2 | Yes | |
RAPDCBCRJCIZDZ
|
8.5 | IC50 | 2 | — | |
HPCDTQWLMQWOIN
|
8.5 | IC50 | 2 | — | |
FDGCWUJGJDWRLS
|
8.5 | IC50 | 2 | — | |
INTUFYOHDOYBRZ
|
8.3 | IC50 | 2 | — | |
VKQZQIDNZZTHCQ
|
8.3 | IC50 | 2 | — | |
BBKUNIDRTSPPPW
|
8.2 | Ki | 2 | Yes | |
CIQFRWAEJMYDAF
|
8.2 | IC50 | 2 | — | |
DLVZGEWWOWCZQG
|
8.2 | IC50 | 2 | — | |
CIQDQPSLIUICPX
|
8.2 | IC50 | 2 | — | |
XRYUXASBLSDNDZ
|
8.1 | IC50 | 2 | — |