Target Details
| UniProt AC | P46531 |
|---|---|
| Gene Symbol | NOTCH1 |
| Protein Name | Neurogenic locus notch homolog protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00008 (EGF) PF07645 (EGF_CA) PF12661 (hEGF) PF06816 (NOD) PF07684 (NODP) PF00066 (Notch) |
Summary
- Multi-target molecules 84
- Clinical molecules 0
- Avg pChEMBL 8.32
KEGG Pathways (9)
Associated Diseases (4)
Active Molecules (84)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AHQDKFUMSUHJRJ
|
8.3 | IC50 | 2 | — | |
JDQVYMCRALZOEK
|
8.3 | IC50 | 2 | — | |
PUVNOTSVUAEILD
|
8.3 | IC50 | 2 | — | |
AKEGFLOENKCBST
|
8.3 | IC50 | 2 | — | |
SXYFZXGSGRDRFY
|
8.3 | IC50 | 2 | — | |
JADHURSZAFCXCI
|
8.3 | IC50 | 2 | — | |
VPJBPAOAPXODSK
|
8.3 | IC50 | 2 | — | |
WWSOXWIWFGQZFX
|
8.2 | IC50 | 2 | — | |
OHNOCFPDYZDIHV
|
8.2 | IC50 | 2 | — | |
SWHPGUZTSMXLGG
|
8.2 | IC50 | 2 | — | |
ZIRIDNHDVCSNSH
|
8.2 | IC50 | 2 | — | |
HVLALDWMJAWZQF
|
8.2 | IC50 | 2 | — | |
DBRSXVXJAVHIKP
|
8.2 | IC50 | 2 | — | |
XJDSZSLHQRQHLY
|
8.2 | IC50 | 2 | — | |
GPSAOZZYKLGLJH
|
8.2 | IC50 | 2 | — | |
GQQOKRQIUXMKQD
|
8.2 | IC50 | 2 | — | |
NVAQWNDQKADVMO
|
8.1 | IC50 | 2 | — | |
FSRNLFFSZLWWIK
|
8.1 | IC50 | 2 | — | |
MUUVZWZJMPDNOV
|
8.1 | IC50 | 2 | — | |
SRJNRAQUSAVENA
|
8.1 | IC50 | 2 | — | |
MRDOSSIBKDYGQX
|
8.1 | IC50 | 2 | — | |
MCIWNCZITHCVOD
|
8.1 | IC50 | 2 | — | |
LOWIEMBYDPEZKM
|
8.0 | IC50 | 2 | — | |
TWOYRGKPVVYZKA
|
7.9 | IC50 | 2 | — | |
CEVHLIUGNONVJN
|
7.9 | IC50 | 2 | — | |
NBOUPMNHRXSDBV
|
7.9 | IC50 | 2 | — | |
OTUPLGMOMNWEEM
|
7.9 | IC50 | 2 | — | |
SVOOSDGRCIVKOG
|
7.8 | IC50 | 2 | — | |
HPYFEYKGJCBKKX
|
7.5 | IC50 | 2 | — | |
NFSUDFPUVQNBSA
|
7.4 | IC50 | 2 | — | |
DYNTZUXZTDSIOF
|
7.3 | IC50 | 2 | — | |
RTMFXQXENIODOP
|
7.2 | IC50 | 8 | — | |
WGYNBTCNYOMMNG
|
6.8 | IC50 | 2 | — | |
RMRHTXFKXWUOFV
|
6.6 | IC50 | 2 | — |