Target Details
| UniProt AC | P46531 |
|---|---|
| Gene Symbol | NOTCH1 |
| Protein Name | Neurogenic locus notch homolog protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF00008 (EGF) PF07645 (EGF_CA) PF12661 (hEGF) PF06816 (NOD) PF07684 (NODP) PF00066 (Notch) |
Summary
- Multi-target molecules 84
- Clinical molecules 0
- Avg pChEMBL 8.32
KEGG Pathways (9)
Associated Diseases (4)
Active Molecules (84)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BJFMDMZPJSKEEF
|
9.0 | IC50 | 2 | — | |
SMTPPNKOJYQIIG
|
9.0 | IC50 | 2 | — | |
XMSPXAZZQLYGPP
|
9.0 | IC50 | 2 | — | |
UGHSMELYSLKUPL
|
8.8 | IC50 | 2 | — | |
DFPGVOULJBAUOC
|
8.8 | IC50 | 2 | — | |
SDVKHWCDJLBDAQ
|
8.8 | IC50 | 2 | — | |
VVCCUNLSKGRBBX
|
8.8 | IC50 | 2 | — | |
NXOSJQJBUYUAKD
|
8.7 | IC50 | 2 | — | |
AXDPFPZUTDRTAU
|
8.7 | IC50 | 2 | — | |
CMVFMWZCQMQNSS
|
8.7 | IC50 | 2 | — | |
QOSWTKQCJJCHLE
|
8.7 | IC50 | 2 | — | |
SXLRLXYEBHFPKN
|
8.7 | IC50 | 2 | — | |
XGTZKVXMDSWEOE
|
8.7 | IC50 | 7 | — | |
QHRXWPSDABHYNR
|
8.7 | IC50 | 2 | — | |
IALGOODQMCARJD
|
8.6 | IC50 | 2 | — | |
KYAKIRYXKXSQLN
|
8.6 | IC50 | 2 | — | |
ZTPQNQNCCURRQX
|
8.6 | IC50 | 2 | — | |
ISPSTDXOYVVQCC
|
8.6 | IC50 | 2 | — | |
JDPJHJXWAWWFPR
|
8.6 | IC50 | 2 | — | |
SPTBWGHFYWWLSW
|
8.6 | IC50 | 2 | — | |
OXUKVUCQWJCSLA
|
8.5 | IC50 | 2 | — | |
PNAKCIOOKPJNCG
|
8.5 | IC50 | 2 | — | |
AXUCGPSYXKJACT
|
8.5 | IC50 | 8 | — | |
CRNVUALZNXEPSA
|
8.5 | IC50 | 2 | — | |
DGNPZFFWUMSXJB
|
8.5 | IC50 | 2 | — | |
GKQMFTFKNTUDIV
|
8.5 | IC50 | 2 | — | |
HDJFGDOVVAHZMZ
|
8.5 | IC50 | 2 | — | |
JLJBRBHIPOCFTJ
|
8.5 | IC50 | 2 | — | |
XHVDMEMANOFVOM
|
8.5 | IC50 | 2 | — | |
HDBIKHIYDCBTHE
|
8.5 | IC50 | 2 | — | |
VPJBPAOAPXODSK
|
8.5 | IC50 | 2 | — | |
RCLWNQQLQHLLBS
|
8.5 | IC50 | 2 | — | |
HUWDWVSWYJEMFI
|
8.5 | IC50 | 2 | — | |
HMKRFXHMAJMWSE
|
8.5 | IC50 | 2 | — | |
BQJHUPVEKBVMDC
|
8.4 | IC50 | 2 | — | |
WJCNQWZOWZRWNV
|
8.4 | IC50 | 2 | — | |
JULHDMBKEVNXLX
|
8.4 | IC50 | 2 | — | |
NVACINZDYAXFIA
|
8.4 | IC50 | 2 | — | |
SKRPANNVXVGYFB
|
8.4 | IC50 | 2 | — | |
DPJSWEWXBIYMHC
|
8.4 | IC50 | 4 | — | |
VNCVKYZPDLZSFH
|
8.4 | IC50 | 2 | — | |
RGDQPBKNPHAJES
|
8.4 | IC50 | 2 | — | |
HDKLJEMMROHEMQ
|
8.4 | IC50 | 2 | — | |
NKEZCYOXWCSOAX
|
8.4 | IC50 | 2 | — | |
SBOWAFOVKLYUOM
|
8.4 | IC50 | 2 | — | |
TUCRSTOAEKKIOP
|
8.4 | IC50 | 2 | — | |
OYVNZMZRYVSNQD
|
8.3 | IC50 | 2 | — | |
KWECVZITGSUXJY
|
8.3 | IC50 | 2 | — | |
RHYJCCNJGSBGBR
|
8.3 | IC50 | 2 | — | |
GYSCHXPQKTXBHJ
|
8.3 | IC50 | 2 | — |