Target Details
| UniProt AC | P46098 |
|---|---|
| Gene Symbol | HTR3A |
| Protein Name | 5-hydroxytryptamine receptor 3A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 382
- Clinical molecules 7
- Avg pChEMBL 7.39
KEGG Pathways (3)
Active Molecules (382)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PDOCNPCPPLPXRV
|
6.1 | Ki | 5 | — | |
GEKVZXHRWKQTBA
|
6.1 | Ki | 4 | — | |
VZNBEHZTGROPAO
|
6.1 | Ki | 2 | — | |
GNIBIBLEGLWUTE
|
6.1 | Ki | 2 | — | |
OTVQCHUIPJYASM
|
6.1 | Ki | 4 | — | |
CFHPNABTZSOBQJ
|
6.1 | Ki | 5 | — | |
UPQDSOGWDXPNJO
|
6.1 | Ki | 2 | — | |
DZSVIKVOAPBNLM
|
6.1 | Ki | 5 | — | |
ZRPDKOIUHULZCY
|
6.1 | Ki | 7 | — | |
BDLSNMGOWYNTSL
|
6.1 | Ki | 3 | — | |
CKDXPZFNUORSGK
|
6.1 | Ki | 2 | — | |
ILEIGUXOYKZHRK
|
6.0 | Ki | 5 | — | |
TXFAZGWNVUZLNN
|
6.0 | Ki | 2 | — | |
HIFHKIVBOAYGIT
|
6.0 | Ki | 2 | — | |
WECKJONDRAUFDD
|
6.0 | Ki | 2 | — | |
AGJYNAQBTFSPHI
|
6.0 | Ki | 2 | — | |
AJTVQZWUKUPHIP
|
6.0 | IC50 | 3 | — | |
BKVIWGRFRKLFIO
|
6.0 | Ki | 9 | — | |
DICVBGGIAAPPNV
|
6.0 | Ki | 3 | — | |
GROYHNLGVCIQOI
|
6.0 | Ki | 8 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
IEUXRHDPSSNADT
|
6.0 | Kd | 5 | — | |
KAJKLJPCBJPNMB
|
6.0 | Ki | 2 | — | |
LOCQRDBFWSXQQI
|
6.0 | Ki | 16 | — | |
OKGUIDHKHQYCQC
|
6.0 | Ki | 2 | — | |
QLOOWOVVZLBYHU
|
6.0 | Ki | 7 | — | |
QQJHRQZZCNYDMX
|
6.0 | Ki | 11 | — | |
SWEOAXMICIJCQC
|
6.0 | Ki | 4 | — | |
VGFALHATLLBXIT
|
6.0 | Ki | 5 | — | |
VHGCDTVCOLNTBX
|
6.0 | Ki | 19 | — | |
YOGJZQGRTVMCPY
|
6.0 | IC50 | 17 | — | |
ZZZQXCUPAJFVBN
|
6.0 | Ki | 7 | — |