Target Details
UniProt ACP46098
Gene SymbolHTR3A
Protein Name5-hydroxytryptamine receptor 3A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 382
  • Clinical molecules 7
  • Avg pChEMBL 7.39
Top Co-occurrence Targets
Active Molecules (382)
InChIKey pChEMBL Type Targets Clinical
PNROIWQNPITPBR 6.4 Ki 5
SVFXJOTZHCGIKP 6.4 Ki 2
KSGSFRSZNPFDNI 6.4 Ki 2
OFHWWCZOJZHPFZ 6.4 Ki 2
PKQYVFHRKFDVCH 6.4 Ki 5
KVWDHTXUZHCGIO 6.3 Ki 32 Yes
OBWCQARWOVVGRJ 6.3 Ki 5
WLVXTRCIWADVNT 6.3 Ki 2
JTLCTTWVUAIQHD 6.3 IC50 17 Yes
WNUBZTJAEYKDQZ 6.3 Ki 2
XJNOJISWTROLSF 6.3 IC50 2
ZDTPXUKLGIDOCS 6.3 IC50 2
GQPFOKFRIDVKLE 6.3 Ki 4
RCCDDPHPJBBTOH 6.3 Ki 4
UVOCSZKGWJOKNN 6.3 Ki 11
LGWFAAILRNJWJB 6.3 Ki 6
MMSIHQRSTJAVNZ 6.2 Ki 6
QLADKQSPDYCWLO 6.2 Ki 3
VYZPEWUEPPGXGA 6.2 Ki 5
HIWIXUJADKOVEP 6.2 Ki 2
IPKZCLGGYKRDES 6.2 Ki 6
UKSIPAJWYFDSNE 6.2 Ki 2
ALRBWNXPNRLJKC 6.2 Ki 10
JOIYZVWBZFRJTG 6.2 IC50 2
ORMRVPRSUUACQQ 6.2 Ki 3
UZJWAFOJOSGEKL 6.2 IC50 15
YQBFPVBTXMITDN 6.2 Ki 2
CXDMUUBLDHSHNL 6.2 Ki 6
IPZJPIUIHUHJMB 6.2 Ki 2
WSKZCTVUXTXPQV 6.2 Ki 2
YVENIGOVHPMTDH 6.2 Ki 23
IEXWVCPGJPZNIH 6.2 Ki 2
JBPBJYKHTQKMKP 6.2 Ki 4
ALPVAQHXSGKIAL 6.2 Ki 6
BGMSTNYJYPSLHN 6.2 IC50 4
DFPVYCZMZZRMKO 6.2 Ki 2
HDVMGKGTLCDZNU 6.2 Ki 2
IQJBDRJDMXGXFH 6.2 Ki 3
RYBOXBBYCVOYNO 6.2 Ki 10
XBNNPPLRTCDVRJ 6.2 Ki 4
CZXYEUKDTXJZAI 6.2 Ki 2
MREMSPSMZSVSJS 6.2 Ki 3
GTUIQNHJSXQMKW 6.2 Ki 3
JKXJYPUQCHXWQU 6.2 Ki 2
RHFLZSUIVOSCKT 6.2 Ki 6
CEUORZQYGODEFX 6.2 Ki 31
KMWRABRPTOODHP 6.2 Ki 4
QWJGFXHJEQDQOM 6.2 IC50 2
ZUCQKAOSMQWPJG 6.2 Ki 5
MJJDYOLPMGIWND 6.1 Ki 5
2D structure