Target Details
UniProt ACP46098
Gene SymbolHTR3A
Protein Name5-hydroxytryptamine receptor 3A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 382
  • Clinical molecules 7
  • Avg pChEMBL 7.39
Top Co-occurrence Targets
Active Molecules (382)
InChIKey pChEMBL Type Targets Clinical
HKPHVFFQXHMOHX 6.7 Ki 5
HTYFFCPFVMJTKM 6.7 Ki 5
OKBKFPZFYXEZPA 6.7 Ki 2
YMMFEXFJXKPQGZ 6.7 Ki 2
ZXTPPBDZBKAHMV 6.7 Kd 5
BRNUKIDBYPCLGD 6.7 IC50 5
DNJXPDYLZIVHDP 6.7 IC50 5
IWXFOGIXCQWSGX 6.7 Ki 2
WEOIHIYCKWSSBW 6.7 Ki 5
CDUXPGVKEOGWKB 6.7 IC50 2
LIIRNJNGOKYCIP 6.7 Ki 5
DMGKTIDNNWALJM 6.6 Ki 2
IUNFWMWQNWQIFS 6.6 Ki 5
JIGWWGDIEUWCOR 6.6 Ki 5
YSCNOWHLCXMNDZ 6.6 Ki 3
DTOKLFDSWKGLOX 6.6 Ki 5
PKWXICSBZZLGCF 6.6 Ki 2
UVEYNCQCHBIENE 6.6 Ki 2
BTTOYOKCLDAHHO 6.6 Ki 10
CCGSTBSDYHGTEC 6.6 Ki 2
HRWKDXOKUOFVIB 6.6 Ki 2
HRWKDXOKUOFVIB 6.6 Ki 2
JJNKQQZKWYVYGT 6.6 Ki 2
OZINHCFSCQEUPW 6.6 Ki 5
DFGJMJURTZFUDF 6.5 Ki 2
VFIFSUHWHJHYJR 6.5 Ki 2
YJNPVKYWRQNPBX 6.5 IC50 5
CDBWVULDFPANMP 6.5 Ki 2
IYYKRUUXDACSBG 6.5 Ki 5
QYUZYZBBJGTSFR 6.5 Ki 6
SSRDSYXGYPJKRR 6.5 IC50 2
MUOXAGUZMVATIC 6.5 Ki 2
OBSQXMOZMFTQSH 6.5 Ki 2
ZSJNJAJDBNFVCA 6.5 Ki 5
UFXJIPGDVROFEN 6.5 Ki 2
HETPCFGGOCHPAU 6.5 IC50 2
ZCVMWBYGMWKGHF 6.5 Ki 19 Yes
DJKJVWJQAVGLHJ 6.5 Ki 8
GMRSWLGFTCTQFO 6.4 Ki 2
HXPQWNPLNIEJOW 6.4 Ki 3
RKFZJZNWZIIGFB 6.4 Ki 2
ZSVHQGYEWBPZFU 6.4 Ki 2
MVWVFYHBGMAFLY 6.4 Ki 31 Yes
RZBUCINSAXOVJU 6.4 Ki 2
GDRLBCZDGQFDCZ 6.4 Ki 7
NKPRIPDEFRADKU 6.4 Ki 6
ZINGRQZUIVEPKX 6.4 Ki 2
AJUQPEHETMTGCL 6.4 Ki 2
HZUVTGUCSFHZGQ 6.4 Ki 7
MQLWANLDQKRYQY 6.4 Ki 8
2D structure