Target Details
UniProt ACP46098
Gene SymbolHTR3A
Protein Name5-hydroxytryptamine receptor 3A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 382
  • Clinical molecules 7
  • Avg pChEMBL 7.39
Top Co-occurrence Targets
Active Molecules (382)
InChIKey pChEMBL Type Targets Clinical
IRNHNTVMAZMVND 7.2 Ki 2
ZHSLKEYCKRMUKN 7.2 Ki 2
XOUOEUATRAFRCX 7.2 Ki 5
ZSDSOMKIKNSFJG 7.2 Ki 3
HLMKBCUKQMBYDR 7.2 IC50 2
HNDKJDCYXITJAR 7.2 Ki 5
PKPRDSSAMMLSLJ 7.2 IC50 2
ZIZADASDJMYXQQ 7.2 Ki 2
OFXSSUCHCSBXFS 7.1 Ki 3
OMACXBJTMXFHCQ 7.1 IC50 2
BPUACIBQBJYAPM 7.1 Ki 2
LCGYRMCRRGNDFQ 7.1 Ki 2
QBSLBAVTMNFTOR 7.1 Ki 2
ZSTKHSQDNIGFLM 7.1 Kd 22
CAIDHVXIMVKUTP 7.1 Ki 2
UXDSQRDGBDALMX 7.1 Ki 2
DEMZYMHKNNMIGU 7.1 IC50 5
PXAINPSPSFFTMA 7.1 IC50 5
YZHWETPHARDZQM 7.1 IC50 2
MDDLXKDIADSAQA 7.0 IC50 2
YLVNDFYGPNTLDN 7.0 Ki 2
WPVVMKYQOMJPIN 7.0 Ki 5
BOJVRMCXKCSTBM 7.0 Ki 2
FRVUAAGRCGXHSZ 7.0 Ki 2
NLWMJOOAJCUQKB 7.0 Ki 2
ARCIIEQRTPPAQU 6.9 IC50 5
FFNWMBDISAYHDC 6.9 Ki 2
PDTVBRINWYWWLT 6.9 Ki 5
FBDSJUSEZSFHOW 6.9 Ki 2
ONIODQRFDDUVAG 6.9 Ki 2
QZAYGJVTTNCVMB 6.9 Ki 17
OMMHQUDWONZRDG 6.8 Ki 2
QKWNDCGZOXJVDP 6.8 Ki 2
AXKDMCQUCRBQFP 6.8 Ki 5
DCSUBABJRXZOMT 6.8 Kd 24
GAYSOZKZPOVDSB 6.8 Ki 5
GTMRUYCIJSNXGB 6.8 Ki 2
GTMRUYCIJSNXGB 6.8 Ki 2
OFXSSUCHCSBXFS 6.8 Ki 3
UJNJZDZUOJYRAQ 6.8 Ki 2
UQSXOKQEMNCJCE 6.8 Ki 2
GGBKKIVDGBAYTK 6.8 Ki 2
DIBHIFSZXTZWAW 6.8 Ki 2
VBKOTIVQMCTTAQ 6.8 Ki 5
VNICFCQJUVFULD 6.8 Ki 15
AOOSJYIINXVNHV 6.8 Ki 16
AFLJKKMTBWNZFE 6.7 Ki 6
IXUOQYGGXPUKBV 6.7 Ki 2
XFTKDUCZMYGGEC 6.7 Ki 2
QZUDBNBUXVUHMW 6.7 Ki 39 Yes
2D structure