Target Details
UniProt ACP46098
Gene SymbolHTR3A
Protein Name5-hydroxytryptamine receptor 3A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 382
  • Clinical molecules 7
  • Avg pChEMBL 7.39
Top Co-occurrence Targets
Active Molecules (382)
InChIKey pChEMBL Type Targets Clinical
AOWDEXMOARHNIR 7.5 Ki 2
DWLMIHRZURMFAQ 7.5 Ki 5
LWLBVIFUVSUSAY 7.5 Ki 6
MBWUFSQDLZYQLA 7.5 Ki 2
OUENCNZMGZDHGX 7.5 Ki 2
KOCIMJYSVMTYIG 7.5 Ki 2
BPPGPYJBCVXILI 7.5 IC50 5
KIJXVALDJPUIFM 7.5 Ki 6
LDIYRDXQPDSEFR 7.5 IC50 5
HASGWVOTHYCRIP 7.4 Ki 5
LQLAPWUVEHKEPV 7.4 Ki 2
NGQQPARRDBDNPB 7.4 Ki 3
KIVOPFOXJNXWFW 7.4 Ki 5
OOMBBUZQJGYRRW 7.4 Ki 5
FCZBQMUDGBEIHG 7.4 Ki 5
JZSPAHAWDCQCEX 7.4 Ki 5
DAZOPYDOJHNKSD 7.4 Ki 5
NWVOTDQIZMJKRJ 7.4 Ki 5
DFGJMJURTZFUDF 7.4 Ki 2
ZQJXKMUGFKJVKD 7.4 Ki 2
SDFWQNVGYRAAAZ 7.3 Ki 5
FMWXWOAWFBYPCO 7.3 IC50 5
QZEXFNKCPOFGAE 7.3 Ki 2
BMIQQALNTAJMLB 7.3 Ki 5
HIQWVKZIJAMSHI 7.3 Ki 2
VWVPNALHKWLANG 7.3 IC50 2
MYBMSIDXODXJBU 7.3 IC50 2
SSOHJAKQLOENEM 7.3 Ki 6
TTWJBBZEZQICBI 7.3 Kd 10
FZGWDCDUMFWUEO 7.3 IC50 9
DQFJTXJCMDYWKL 7.3 IC50 2
FBFVECUFQXIPMF 7.3 Ki 3
FGDWUDRNOXESRS 7.3 Ki 2
JXOLMXLINBXECI 7.3 Ki 5
QKMVBIUHVBVHGX 7.3 Ki 2
XXJMPUMRHCNWPW 7.3 Ki 8
UGLUCZYCHYWOCD 7.3 IC50 2
HAMAPMMCMQNNBY 7.2 Ki 2
UMHNYWDDWJWNHJ 7.2 Kd 5
FXKDRFDFQGJXIQ 7.2 IC50 2
GGDBEAVVGFNWIA 7.2 Ki 6
XFRTZUYXJVAJNT 7.2 Ki 5
ABSDJNLAUZQHJY 7.2 Ki 2
MKWFJPZMYHPQIA 7.2 Ki 5
VHFVKMTVMIZMIK 7.2 Ki 15
HMOMXYPGOQVVIY 7.2 Kd 5
LGKSUDPSBCMQRR 7.2 Ki 5
OJNSMLDRVFFVJN 7.2 IC50 2
PCWGGOVOEWHPMG 7.2 Ki 12
XQJMXPAEFMWDOZ 7.2 Kd 5
2D structure