Target Details
UniProt ACP46098
Gene SymbolHTR3A
Protein Name5-hydroxytryptamine receptor 3A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 382
  • Clinical molecules 7
  • Avg pChEMBL 7.39
Top Co-occurrence Targets
Active Molecules (382)
InChIKey pChEMBL Type Targets Clinical
QNKGTIWNFNPEJL 8.1 IC50 11
SSQNUJKKRPIPQK 8.1 Kd 5
SFVKVHVOODTRCH 8.1 Ki 2
SFVKVHVOODTRCH 8.1 Ki 2
WZYBXWXOBIOGBH 8.1 Ki 5
KQKPFRSPSRPDEB 8.0 IC50 9
BOHGZALGHLQJNA 8.0 IC50 7
ATJCEXDPRCAAOP 8.0 Ki 5
QENBLMVKRYFDIR 8.0 IC50 5
GIRLVGYIIVFTLI 7.9 Ki 6
OCKIPDMKGPYYJS 7.9 Ki 4
PELIXYXPUAFHOR 7.9 Ki 2
RDLIBCPWPNCFBW 7.9 Ki 5
SECBCZUIMWWSPE 7.9 Ki 2
XYOILXJZQNPSEP 7.9 IC50 7
YQNWZWMKLDQSAC 7.9 Ki 15
ZJAWVBLMRPEUPW 7.9 Ki 5
FKFNPTZCZKTCNF 7.9 Ki 2
CXJLWJAYGMWLRR 7.9 Ki 2
JUSBDZIBILCYFG 7.9 IC50 5
CBXQAAQVKDTXJJ 7.9 Ki 2
SXXANLLRNHHDSR 7.8 IC50 5
XGEHMWGDEOZVML 7.8 IC50 5
AUISQHXDGNJFJZ 7.8 Ki 5
BQFFJFYYLYTLCC 7.8 Ki 2
OZOLNJQERDKPFN 7.8 Ki 2
OZOLNJQERDKPFN 7.8 Ki 2
KQFRTJUIRPBBAB 7.8 Ki 5
DIHXJZHAIHGSAW 7.8 Ki 5
QNJWNYDKHQYCPI 7.8 Ki 2
SOEFWQWHKHCTLH 7.7 IC50 2
PXSRGUBKHGVLLK 7.7 Ki 5
AYDBLCSLKNTEJL 7.7 Kd 5
BUOWEEIISDGZDM 7.7 IC50 5
ILDJOTZORZWBSP 7.7 IC50 5
YMQVTFAERCACRG 7.7 IC50 5
UNLXJJLVSBLRLU 7.7 Ki 5
XGSROJUGJKXEPW 7.6 IC50 5
UVZMYAXDXQFDBO 7.6 IC50 5
OHXKHPFEXVDLQZ 7.6 IC50 2
SGKHROGKIKKECN 7.6 Ki 5
OKFGYYBZAZENKT 7.6 Ki 2
QHJZTYYNXIQQNW 7.6 Ki 3
RYAZLYGDKFCFKI 7.6 Ki 2
XQMDXRYDYUXFEH 7.5 Ki 5
YVTHPCKJOKJJHA 7.5 IC50 5
FEPRMAUTVAUZGM 7.5 IC50 5
IFZNYQPTDBKBSE 7.5 Ki 2
YYXITPMMGBMZSU 7.5 Ki 2
VQMVUGKLGFORBP 7.5 IC50 5
2D structure